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Chemicals & Small Molecules

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    Results for Chemicals & Small Molecules ( 97581 )

      • ANR 94

        Ref: T22031
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: DKK300.00

        ANR 94 (Legacy Tebubio ref. 282T22031). ANR94 is a potent, selective antagonist of the adenosine A2A receptor (AA2AR), exhibiting a K_i value of 46 nM for the human AA2AR (hAA2AR). This compound shows promise for research into Parkinson's disease. [1] [2]

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      • ARC 239 dihydrochloride

        Ref: T22033
        Sizes: 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: DKK293.00

        ARC 239 dihydrochloride (Legacy Tebubio ref. 282T22033). ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist with pKD values of 8.8, 6.7, and 6.4 at α2B, α2A, and α2D receptors respectively (pKD values are 8.8, 6.7, and 6.4 at α2B, α2A, and α2D receptors respectively).

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      • ARP 101

        Ref: T22034
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: DKK855.00

        ARP 101 (Legacy Tebubio ref. 282T22034). ARP 101 is an effective selective matrix metalloproteinase-2 (MMP-2) inhibitor with anti-cancer activity. It induces the inhibition of HCMV through non-classical chelate 1 (SQSTM1)/p62-Keap1-Nrf2 pathways and phosphorylation of the C-terminal domain of p62, regulating autophagy and inhibiting melanogenesis.

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      • Arylquin 1

        Ref: T22036
        Sizes: 1 mg, 5 mg, 10 mg
        From: DKK668.00

        Arylquin 1 (Legacy Tebubio ref. 282T22036). Arylquin 1, a prostate-apoptosis-response-4 (Par-4) secretagogue, specifically targets vimentin to facilitate Par-4 secretion. It also induces lysosomal membrane permeabilization (LMP) and promotes non-apoptotic cell death in cancer cells [1].

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      • AS 1892802

        Ref: T22037
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: DKK375.00

        AS 1892802 (Legacy Tebubio ref. 282T22037). AS 1892802 is a potent and selective inhibitor of ROCK. AS 1892802 exibits IC50 values of 52nM, 57nM and 122 nM for human ROCK2, rat ROCK2 and human ROCK1, respectively. The onset of antinociceptive effect of AS 1892802 is as fast as those of Tramadol and Diclofenac.

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      • Diaveridine

        Ref: T2204
        Sizes: 1 g, 500 mg, 1 mL * 10 mM (in DMSO)
        From: DKK263.00

        Diaveridine (Legacy Tebubio ref. 282T2204). Diaveridine (AI3-23935) (DVD) is a popular antibacterial synergist that is widely used in combination with sulfonamide. It has been reported to be genotoxic to mammalian cells, but more studies are required to clarify this.

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      • BCATc Inhibitor 2

        Ref: T22043
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: DKK435.00

        BCATc Inhibitor 2 (Legacy Tebubio ref. 282T22043). BCATc Inhibitor 2 exhibited an IC50 of 0.8 microM in the hBCATc assays; it is an active and selective inhibitor. BCATc Inhibitor 2 also blocked calcium influx into neuronal cells following inhibition of glutamate uptake, and demonstrated neuroprotective efficacy in vivo[1]. Branched-chain amino acid transferases (BCATs) have been implicated in catalyzing reversible transamination of isoleucine, leucine, and valine branched-chain amino acids to their corresponding α-keto acids, generating L-glutamate. It has been identified that there are two forms of BCAT in mammals: mitochondrial BCAT (BCATm) and cytosolic BCAT (BCATc). BCATc is expressed in particular brain region and involved in regulating glutamate synthesis for release during neuronal excitation. Thus, BCATc inhibition may be useful for the treatment of neurodegenerative and behavioral disorders involving disturbances of the glutamatergic system [2].

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      • BGC 20-761

        Ref: T22044
        Sizes: 10 mg
        From: DKK4,928.00

        BGC 20-761 (Legacy Tebubio ref. 282T22044). BGC20-761 is a selective 5-HT6 and dopamine receptor antagonist (human receptor K i values: 5-HT6 (20 nM), 5-HT2A (69 nM), D2 (140 nM)), and a tryptamine analog with a high affinity for 5-HT(6) receptors, that can enhance long-term memory, with potential utility as an antipsychotic agent [1].

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      • bis(7)-Tacrine

        Ref: T22048
        Sizes: 5 mg, 100 mg, 10 mg
        From: DKK1,688.00

        bis(7)-Tacrine (Legacy Tebubio ref. 282T22048). Bis(7)-tacrine dihydrochloride is a dimeric AChE inhibitor derived from tacrine with potential to treat Alzheimer's disease, prevents glutamate-induced neuronal apoptosis by blocking NMDA receptors, and is a potent GABA A receptor antagonist[1] [2] [3].

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