KKI-5 acetate(97145-43-2 free base) (Legacy Tebubio ref. 282TP1792L). KKI-5 acetate is a serine protease inhibitor that inhibits kallikrein and plasmin. KKI 5 may exhibit anticancer chemotherapeutic benefit and may also be used as a treatment for angioedema.
Nociceptin (1-13), amide (Legacy Tebubio ref. 282TP1793). Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist, exhibiting a pEC50 of 7.9 in mouse vas deferens and a Ki of 0.75 nM for rat forebrain membrane binding.
Nociceptin (1-13) amide TFA (Legacy Tebubio ref. 282TP1793L). Nociceptin (1-13), amide is a potent agonist Opioid receptor-like1 (ORL1) receptor with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain membranes.
S961 (Legacy Tebubio ref. 282TP1795). S961 is a high-affinity, selective insulin receptor (IR) antagonist with IC50 values of 0.048 nM for HIR-A, 0.027 nM for HIR-B, and 630 nM for human insulin-like growth factor I receptor (HIGF-IR) in scintillation proximity assays.
Albiglutide TFA (782500-75-8 free base) (Legacy Tebubio ref. 282TP1796). Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
Pep-1 (uncapped) (Legacy Tebubio ref. 282TP1798). Pep-1 (uncapped), which has 21 amino acid residues, is a known carrier peptide that delivers full-length native proteins in vitro and in vivo.
Z-Gly-Gly-Arg-AMC (Legacy Tebubio ref. 282TP1799). Z-Gly-Gly-Arg-AMC is a specific fluorogenic substrate used to assess thrombin generation and thrombin activity in Platelet-Rich Plasma (PRP) and Platelet-Poor Plasma (PPP).
pGlu-Pro-Arg-MNA (Legacy Tebubio ref. 282TP1800). pGlu-Pro-Arg-MNA [N-(3-[2-Furyl]-acryloyl) - L - leucyl - glycyl - p - nitroanilide] is a chromogenic peptide substrate, specifically utilized for its role in biochemical assays.
pGlu-Pro-Arg-MNA monoacetate (Legacy Tebubio ref. 282TP1801). pGlu-Pro-Arg-MNA monoacetate, a thrombin substrate modeled after a thrombin cleavage site in human fibrinogen, can be used for sensitive assays of antithrombin III activity.