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    Results for Chemicals & Small Molecules ( 97553 )

      • Ref: TP1885
        Sizes: 1 mg

        [(pF)Phe4]Nociceptin(1-13)NH2 (Legacy Tebubio ref. 282TP1885). Highly potent and selective nociceptin/orphanin FQ receptor (OP4) agonist peptide (pKi = 10.68; pEC50 = 9.80). Displays > 8000-fold selectivity over δ, κ, and μ opioid receptors and has relatively long lasting pronociceptive, hypotensive, negative inotropic and feeding stimulation effects in vivo.

        Product detail
      • Ref: TP1885L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg
        From: DKK2,790.00

        [(pF)Phe4]Nociceptin(1-13)NH2 acetate (Legacy Tebubio ref. 282TP1885L1). [(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31. [(pF)Phe4]Nociceptin(1-13)NH2 acetate displays high selectivity over δ, κ, and μ opioid receptors (>3000 fold).

        Product detail
      • Ref: TP1886L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg
        From: DKK1,133.00

        NoxA1ds acetate(1435893-78-9 free base) (Legacy Tebubio ref. 282TP1886L1). NoxA1ds acetate is a potent and selective NADPH oxidase 1 (NOX1) inhibitor (IC50 : 20 nM). Exhibits selectivity for NOX1 over NOX2, NOX4, NOX5 and xanthine oxidase. Inhibits NOX1-derived O2- production in HT-29 human colon cancer cells. Attenuates VEGF-induced human pulmonary artery endothelial cell migration under hypoxic conditions in vitro.

        Product detail
      • Ref: TP1887
        Sizes: 1 mg

        [Ala107]MBP(104-118) (Legacy Tebubio ref. 282TP1887). Synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 46 - 145 mM).

        Product detail
      • Ref: TP1887L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: DKK2,535.00

        [Ala107]-MBP (104-118) acetate (Legacy Tebubio ref. 282TP1887L1). [Ala107]-MBP (104-118) acetate ([Ala107]-MBP ) is synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 46 - 145 mM).

        Product detail
      • Ref: TP1888
        Sizes: 1 mg

        [Ala113]MBP(104-118) (Legacy Tebubio ref. 282TP1888). Synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 28 - 62 mM).

        Product detail
      • Ref: TP1888L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK1,523.00

        [Ala113]-MBP (104-118) acetate (Legacy Tebubio ref. 282TP1888L1). [Ala113]MBP(104-118) acetate is an noncompetitive peptide inhibitors of protein kinase C (PKC), with IC50s ranging from 28-62 μM.

        Product detail
      • Ref: TP1889
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK1,005.00

        MCL0020 (Legacy Tebubio ref. 282TP1889). MCL0020 is a potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115, and >10,000 nM at MC4, MC3, and MC1 receptors, respectively). It significantly reverses stress-induced anorexia without affecting food intake in free-feeding rats and exhibits anxiolytic-like activity in vivo.

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      • Ref: TP1890
        Sizes: 1 mg, 5 mg, 10 mg, 500 μg
        From: DKK668.00

        MLCK inhibitor peptide 18 (Legacy Tebubio ref. 282TP1890). Selective competitive inhibitor of myosin light chain kinase (IC50 = 50 nM). Displays 4000-fold selectivity over CaM kinase II and does not inhibit PKA. Cell permeable.

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