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    Results for Chemicals & Small Molecules ( 97553 )

      • Ref: TP1901L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK2,108.00

        Hemopressin (rat) acetate(568588-77-2 free base) (Legacy Tebubio ref. 282TP1901L1). Hemopressin (rat) acetate is a nonapeptide derived from the α1-chain of hemoglobin, is originally isolated from rat brain homogenates. Hemopressin is orally active, selective and inverse agonist of CB2 cannabinoid receptors. Hemopressin exerts antinociceptive action in inflammatory pain models.

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      • Ref: TP1902
        Sizes: 1 mg

        G-Protein antagonist peptide (Legacy Tebubio ref. 282TP1902). Substance P-related peptide that inhibits binding of G proteins to their receptors. Competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors.

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      • Ref: TP1902L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg
        From: DKK1,185.00

        G-Protein antagonist peptide acetate (Legacy Tebubio ref. 282TP1902L1). G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide acetate inhibits the activation of Gi or Go by M2 muscarinic cholinergic receptor (M2 mAChR) or of Gs by beta-adrenergic receptor in the reconstituted phospholipid vesicles, assayed by receptor-promoted GTP hydrolysis

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      • Ref: TP1903
        Sizes: 1 mg, 5 mg
        From: DKK1,223.00

        PKG inhibitor peptide (Legacy Tebubio ref. 282TP1903). Competitive inhibitor of cGMP-dependent protein kinase (PKG); analog of a substrate peptide corresponding to a phosphorylation site of histone H2B. Competes with synthetic substrates (Ki = 86 mM) but does not inhibit phosphorylation of intact histones by PKG. Inhibits phosphorylation of intact histones by PKA.

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      • Ref: TP1904
        Sizes: 1 mg, 5 mg, 25 mg, 10 mg
        From: DKK1,905.00

        FSLLRY-NH2 (Legacy Tebubio ref. 282TP1904). Selective PAR2 peptide antagonist. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice. Blocks ERK activation and collagen production in isolated cardiac fibroblasts. Also reduces symptoms in a mouse model of dermatophyte-associated itch.

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      • Ref: TP1904L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg
        From: DKK840.00

        FSLLRY-NH2 TFA(245329-02-6 free base) (Legacy Tebubio ref. 282TP1904L). FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice. Blocks ERK activation and collagen production in isolated cardiac fibroblasts. Also reduces symptoms in a mouse model of dermatophyte-associated itch.

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      • Ref: TP1905
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: DKK338.00

        BW-180C (Legacy Tebubio ref. 282TP1905). BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.

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      • Ref: TP1906
        Sizes: 1 mg

        DPC-AJ1951 (Legacy Tebubio ref. 282TP1906). Potent 14 amino acid peptide agonist of the parathyroid hormone (PTH) receptor (EC50 = 26 nM).

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      • Ref: TP1906L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK1,613.00

        DPC AJ1951 acetate (Legacy Tebubio ref. 282TP1906L1). DPC-AJ1951 acetate, a 14 amino acid peptide that acts as a potent agonist of the parathyroid hormone (PTH)/PTH-related peptide receptor (PPR). And characterized the activity of DPC-AJ1951 acetate in ex vivo and in vivo assays of bone resorption[1].

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