Results for Chemicals & Small Molecules ( 97553 )
- Ref: TP1901L1Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mgFrom: DKK2,108.00
Hemopressin (rat) acetate(568588-77-2 free base) (Legacy Tebubio ref. 282TP1901L1). Hemopressin (rat) acetate is a nonapeptide derived from the α1-chain of hemoglobin, is originally isolated from rat brain homogenates. Hemopressin is orally active, selective and inverse agonist of CB2 cannabinoid receptors. Hemopressin exerts antinociceptive action in inflammatory pain models.
- Ref: TP1902L1Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mgFrom: DKK1,185.00
G-Protein antagonist peptide acetate (Legacy Tebubio ref. 282TP1902L1). G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide acetate inhibits the activation of Gi or Go by M2 muscarinic cholinergic receptor (M2 mAChR) or of Gs by beta-adrenergic receptor in the reconstituted phospholipid vesicles, assayed by receptor-promoted GTP hydrolysis
- From: DKK1,223.00
PKG inhibitor peptide (Legacy Tebubio ref. 282TP1903). Competitive inhibitor of cGMP-dependent protein kinase (PKG); analog of a substrate peptide corresponding to a phosphorylation site of histone H2B. Competes with synthetic substrates (Ki = 86 mM) but does not inhibit phosphorylation of intact histones by PKG. Inhibits phosphorylation of intact histones by PKA.
- From: DKK1,905.00
FSLLRY-NH2 (Legacy Tebubio ref. 282TP1904). Selective PAR2 peptide antagonist. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice. Blocks ERK activation and collagen production in isolated cardiac fibroblasts. Also reduces symptoms in a mouse model of dermatophyte-associated itch.
- Ref: TP1904LSizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mgFrom: DKK840.00
FSLLRY-NH2 TFA(245329-02-6 free base) (Legacy Tebubio ref. 282TP1904L). FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice. Blocks ERK activation and collagen production in isolated cardiac fibroblasts. Also reduces symptoms in a mouse model of dermatophyte-associated itch.
- From: DKK1,613.00
DPC AJ1951 acetate (Legacy Tebubio ref. 282TP1906L1). DPC-AJ1951 acetate, a 14 amino acid peptide that acts as a potent agonist of the parathyroid hormone (PTH)/PTH-related peptide receptor (PPR). And characterized the activity of DPC-AJ1951 acetate in ex vivo and in vivo assays of bone resorption[1].