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    Results for Chemicals & Small Molecules ( 97555 )

      • Ref: TP1927
        Sizes: 1 mg

        d[Leu4,Lys8]-VP (Legacy Tebubio ref. 282TP1927). Selective vasopressin V1B receptor agonist (Ki values are 0.16, 64, 100 and 3800 nM for V1B, oxytocin, V2 and V1A receptors respectively). Displays weak antidiuretic, vasopressor and in vitro oxytocic activities.

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      • Ref: TP1927L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg
        From: DKK338.00

        d[Leu4,Lys8]-VP acetate (Legacy Tebubio ref. 282TP1927L1). d[Leu4,Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respectively. d[Leu4,Lys8]-VP acetate exhibits weak antidiuretic, vasopressor and oxytocic activiti

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      • Ref: TP1928
        Sizes: 1 mg

        [Orn5]-URP (Legacy Tebubio ref. 282TP1928). Urotensin-II (UT) receptor pure antagonist (pEC50 = 7.24). Displays no agonist activity unlike other U-II/URP analogs. Inhibits the action of U-II in the rat aorta ring assay.

        Product detail
      • Ref: TP1928L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK1,523.00

        [Orn5]-URP acetate (Legacy Tebubio ref. 282TP1928L1). [Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP exhibits no agonist activity.

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      • Ref: TP1929
        Sizes: 5 mg

        Saralasin (Legacy Tebubio ref. 282TP1929). Competitive non-selective angiotensin II antagonist.

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      • Ref: TP1929L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: DKK968.00

        Saralasin acetate(34273-10-4 free base) (Legacy Tebubio ref. 282TP1929L1). Saralasin acetate is a Non-selective angiotensin II antagonist.

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      • Ref: TP1930
        Sizes: 1 mg
        From: DKK6,158.00

        Spexin (Legacy Tebubio ref. 282TP1930). Potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galanin receptor 1. Endogenous satiety-inducing peptide; inhibits long chain fatty acid uptake by adipocytes and decreases food consumption in diet-induced obese mice and rats. Attenuates LH secretion in goldfish. Exhibits anxiolytic effects in vivo.

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      • Ref: TP1930L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK990.00

        Spexin acetate(1370290-58-6 free base) (Legacy Tebubio ref. 282TP1930L1). Spexin acetate is a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galanin receptor 1. Endogenous satiety-inducing peptide; inhibits long chain fatty acid uptake by adipocytes and decreases food consumption in diet-induced obese mice and rats. Attenuates LH secretion in goldfish. Exhibits anxiolytic effects in vivo.

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      • [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P (Legacy Tebubio ref. 282TP1931). Broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist for the ghrelin receptor (EC50 = 5.2 nM); diminishes constitutive ghrelin receptor signaling. Also antagonist at tachykinin, bradykinin, CCK and bombesin receptors. Induces apoptosis and inhibits cancer cell growth in vitro.

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