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    Results for Chemicals & Small Molecules ( 97555 )

      • Ref: TP1993
        Sizes: 1 mg
        From: DKK9,030.00

        M617 (Legacy Tebubio ref. 282TP1993). Selective galanin GAL1 receptor agonist (Ki values are 0.23 and 5.71 nM for GAL1 and GAL2 receptors respectively). Enhances food consumption in rats following i.c.v. administration and reduces CAP-induced inflammatory pain.

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      • Ref: TP1993L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK2,430.00

        M617 acetate (Legacy Tebubio ref. 282TP1993L). M617 acetate is a selective agonist of galanin receptor 1 (GAL1). M617 acetate acts through central GAL1, promotes GLUT4 expression, and enhances GLUT4 content in the cardiac muscle of type 2 diabetic rats. The Ki values are 0.23 and 5.71 nM for GAL1 and GAL2, respectively.

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      • Ref: TP1994
        Sizes: 1 mg
        From: DKK9,030.00

        M871 (Legacy Tebubio ref. 282TP1994). Selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM for GAL2 and GAL1 receptors respectively). Blocks the pro-nociceptive effect of GAL2 receptor agonists.

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      • Ref: TP1994L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK2,415.00

        M871 acetate (Legacy Tebubio ref. 282TP1994L). M871 acetate is a selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM at GAL2 and GAL1 receptors, respectively).It blocks pronociceptive effects of GAL2 agonists including AR-M1896.

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      • Ref: TP1995
        Sizes: 1 mg

        MAIT 203 (Legacy Tebubio ref. 282TP1995). Inhibits interaction of APC and Asef (RhoGEF4). Inhibits colorectal cancer cell migration and invasion in vitro.

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      • Ref: TP1996
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: DKK1,943.00

        MCH(human, mouse, rat) (Legacy Tebubio ref. 282TP1996). MCH(human, mouse, rat) is a potent endogenous agonist at melanin-concentration hormone (MCH) receptors (IC50 values are 0.3 and 1.5 nM and EC50 values are 3.9 and 0.1 nM at MCH1 and MCH2 receptors respectively). Increases food intake in vivo.

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      • Ref: TP1997
        Sizes: 1 mg

        [Ala17]-MCH (Legacy Tebubio ref. 282TP1997). Potent melanin-concentrating hormone (MCH) receptor agonist (EC50 values are 17 and 54 nM at MCH1 and MCH2 receptors respectively). Displays some selectivity towards MCH1 over MCH2 (Ki values are 0.16 and 34 nM respectively).

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      • Ref: TP1997L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK1,005.00

        [Ala17]-MCH acetate (Legacy Tebubio ref. 282TP1997L). [Ala17]-MCH acetate is a selective ligand for MCHR1 with a Ki of 0.16 nM and Kd of 0.37 nM(Eu3+ chelate-labeled). [Ala17]-MCH acetate shows selectivity over MCHR2 with Ki of 34 nM.

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      • Ref: TP1999
        Sizes: 5 mg

        MEN 11270 (Legacy Tebubio ref. 282TP1999). Peptide antagonist of the B2 bradykinin receptor (pKi = 10.3); conformationally constrained cyclized analog of HOE 140. Blocks hypotension and bronchoconstriction in vivo. Displays selectivity for B2 over 29 other receptors and ion channels (pIC50 < 5.5).

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