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    Results for Chemicals & Small Molecules ( 97555 )

      • Ref: TP2022
        Sizes: 5 mg

        GR231118 (Legacy Tebubio ref. 282TP2022). Potent neuropeptide Y (NPY) Y1 receptor antagonist (pA2 = 10 and 10.5 at rY1 and hY1, receptors respectively). Also a potent and selective NPY Y4 receptor agonist (pEC50 values are 6.0, 8.6 and 6.1 for rY2, hY4 and rY5 receptors respectively). Suppresses food intake in rats in vivo. Also has affinity for neuropeptide FF (NPFF) receptors in vitro (Ki = 43-73 nM).

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      • Ref: TP2023
        Sizes: 1 mg
        From: DKK10,305.00

        GR 64349 (Legacy Tebubio ref. 282TP2023). Potent and selective tachykinin NK2 receptor agonist (EC50 = 3.7 nM in rat colon). Displays > 1000- and > 300-fold selectivity over NK1 and NK3 receptors respectively. Active in vivo.

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      • Ref: TP2024
        Sizes: 1 mg

        GR 82334 (Legacy Tebubio ref. 282TP2024). Tachykinin NK1 receptor antagonist.

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      • Ref: TP2025
        Sizes: 1 mg
        From: DKK6,968.00

        GRK2i (Legacy Tebubio ref. 282TP2025). GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. Corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.

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      • Ref: TP2026
        Sizes: 1 mg

        GRP (porcine) (Legacy Tebubio ref. 282TP2026). Mammalian bombesin-like peptide neurotransmitter that is an agonist for the gastrin-releasing peptide receptor (GRPR). GRP has been reported to activate GABAergic interneurons in the amygdala leading to increased GABA release and fear suppression in mice in vivo. Also involved in mitogenesis, and GI tract and appetite regulation.

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      • Ref: TP2026L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK1,755.00

        GRP (porcine) acetate (Legacy Tebubio ref. 282TP2026L). GRP (porcine) acetate is the gastrin-releasing peptide extracted from porcine pancreata. GRP (porcine) acetate may have a role in the parasympathetic regulation of endocrine and exocrine secretion from the pig pancreas.

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      • Ref: TP2027
        Sizes: 10 mg

        GaTx2 (Legacy Tebubio ref. 282TP2027). Very high affinity ClC-2 blocker (apparent KD ~ 50 pM). Slows ClC-2 activation and inhibits slow-gating but does not inhibit open ClC-2 channels. Selective for ClC-2 over other ClC family members (ClC-0, ClC-1, ClC-3 and ClC-4), CFTR, GABAC, CaCC and KV1.2.

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      • Ref: TP2028
        Sizes: 1 mg
        From: DKK6,218.00

        Galanin (1-29)(rat, mouse) (Legacy Tebubio ref. 282TP2028). Non-selective galanin receptor agonist (Ki values are 0.98, 1.48 and 1.47 nM for GAL1, GAL2 and GAL3 respectively). Anticonvulsant; prevents the occurrence of full kindled seizures in rats.

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      • Ref: TP2030
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: DKK930.00

        Gastrin I, human (Legacy Tebubio ref. 282TP2030). Gastrin I, human (Gastrin I (human)) is an endogenous peptide produced in the stomach that increases pepsinogen and acid secretion via the CCK2 receptor in the rat.

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