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Chemicals & Small Molecules

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    Results for Chemicals & Small Molecules ( 97553 )

      • Urantide

        Ref: TP2106
        Sizes: 10 mg
        From: DKK2,850.00

        Urantide (Legacy Tebubio ref. 282TP2106). Selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behaves as a partial agonist in a calcium mobilization assay (in CHO cells expressing hUT receptors).

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      • Urantide acetate(669089-53-6 free base)

        Ref: TP2106L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: DKK983.00

        Urantide acetate(669089-53-6 free base) (Legacy Tebubio ref. 282TP2106L). Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behaves as a partial agonist in a calcium mobilization assay (in CHO cells expressing hUT receptors).

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      • TAPI 0

        Ref: TP2107
        Sizes: 1 mg
        From: DKK7,620.00

        TAPI 0 (Legacy Tebubio ref. 282TP2107). ADAM-17 (TACE) and MMP inhibitor; attenuates TNF-α processing. Acts in concert with GM6001 to inhibit Chlamydia trachomatis growth.

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      • Histrelin acetate

        Ref: TP2107L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: DKK683.00

        Histrelin acetate (Legacy Tebubio ref. 282TP2107L). Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It acts on particular cells of the pituitary gland called gonadotropes when present in the bloodstream. Histrelin stimulates these cells to release luteinizing hormone and follicle-stimulating hormone. Thus it is considered a gonadotropin-releasing hormone agonist or GnRH agonist.

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      • TAPI 2

        Ref: TP2108
        Sizes: 1 mg
        From: DKK7,605.00

        TAPI 2 (Legacy Tebubio ref. 282TP2108). ADAM-17 (TACE) and MMP inhibitor (Ki = 120 nM at ADAM-17). Sensitizes cancer stem cells to the lethal effects of 5-FU in vitro. Blocks shedding of TNF-α from cell membranes.

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      • TAT 14

        Ref: TP2109
        Sizes: 1 mg, 5 mg, 25 mg, 10 mg
        Price Enquiry

        TAT 14 (Legacy Tebubio ref. 282TP2109). TAT 14, a 14-mer peptide, is an Nrf2 activator with anti-inflammatory properties. TAT-14 increases Nrf2 protein levels due to targeting the Nrf2 binding site on Keap1, but has no effect on Nrf2 mRNA expression.

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      • AT 14 acetate

        Ref: TP2109L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK855.00

        AT 14 acetate (Legacy Tebubio ref. 282TP2109L). TAT 14 acetate, a 14-mer peptide, is an Nrf2 activator with anti-inflammatory properties. TAT 14 acetate increases Nrf2 protein levels due to targeting the Nrf2 binding site on Keap1, but has no effect on Nrf2 mRNA expression.

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      • TAT-Gap19

        Ref: TP2110
        Sizes: 1 mg
        From: DKK6,473.00

        TAT-Gap19 (Legacy Tebubio ref. 282TP2110). Cx43 hemichannel blocker (IC50 ~7 μM). No significant affinity for gap junctions or Panx1 channels. N-terminal transactivator of transcription (TAT) motif promotes membrane permeability and increases inhibitory effect of Gap19. Active in vivo. Brain penetrant.

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      • TAT-Gap19 acetate

        Ref: TP2110L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK495.00

        TAT-Gap19 acetate (Legacy Tebubio ref. 282TP2110L). TAT-Gap19 acetate is a specific inhibitor of connexin43 hemichannel (Cx43 HC). TAT-Gap19 acetate traverses the blood-brain barrier and alleviates liver fibrosis in mice. TAT-Gap19 acetate does not inhibit the corresponding Cx43 GJCs.

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