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Chemicals & Small Molecules

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    Results for Chemicals & Small Molecules ( 97553 )

      • TAT-GluA2 3Y acetate(1404188-93-7 free base)

        Ref: TP2111L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: DKK1,050.00

        TAT-GluA2 3Y acetate(1404188-93-7 free base) (Legacy Tebubio ref. 282TP2111L). TAT-GluA2 3Y acetate is an inhibitor of AMPA receptor endocytosis.Systemic administration of Tat-GluA2(3Y) during the induction phase of d-amphetamine blocked maintenance of behavioural sensitization and attenuated the maintenance of neurochemical sensitization of rat.

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      • TC14012

        Ref: TP2112
        Sizes: 1 mg
        From: DKK7,028.00

        TC14012 (Legacy Tebubio ref. 282TP2112). CXCR4 antagonist and ACKR3 (CXCR7) agonist (EC50 = 350 nM for CXCR7).

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      • TC14012 acetate

        Ref: TP2112L
        Sizes: 1 mg, 5 mg, 25 mg, 50 mg, 10 mg
        From: DKK660.00

        TC14012 acetate (Legacy Tebubio ref. 282TP2112L). TC14012 acetate is a serum-stable derivative of T140 which is a selective and peptidomimetic CXCR4 antagonist with an IC50 of 19.3 nM. TC14012 is also a potent CXCR7 agonist with an EC50 of 350 nM for recruiting β-arrestin 2 to CXCR7. TC14012 has anti-cancer activity and anti-HIV activity.

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      • Tertiapin LQ

        Ref: TP2113
        Sizes: 10 mg
        Price Enquiry

        Tertiapin LQ (Legacy Tebubio ref. 282TP2113). Blocker of Kir1.1 channels; displays >250-fold selectivity for Kir1.1 (Kd values are 1.1, 274 and 361 nM for Kir1.1, Kir3.1/3.2 and Kir3.1/3.4 respectively). Derivative of tertiapin-Q.

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      • Tertiapin-Q

        Ref: TP2114
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: DKK1,253.00

        Tertiapin-Q (Legacy Tebubio ref. 282TP2114). Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner and inhibits efflux to K(+).

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      • Tertiapin-Q acetate

        Ref: TP2114L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg
        From: DKK1,260.00

        Tertiapin-Q acetate (Legacy Tebubio ref. 282TP2114L). Tertiapin-Q acetate is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner and inhibits efflux to K(+).

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      • SAH-EZH2

        Ref: TP2115
        Sizes: 5 mg
        Price Enquiry

        SAH-EZH2 (Legacy Tebubio ref. 282TP2115). EZH2/EPP interaction inhibitor (Kd = 320 nM). Suppresses EZH2 expression and H3K27 trimethylation by PCR2 complex. Arrests proliferation and induces monocyte to macrophage differentiation of MLL-AF9 leukemia cell line.

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      • SAH-SOS1A

        Ref: TP2116
        Sizes: 5 mg
        Price Enquiry

        SAH-SOS1A (Legacy Tebubio ref. 282TP2116). KRas/son of sevenless 1 (SOS1) interaction inhibitor. Binds within nucleotide binding pocket of KRas (Kd values are 106 - 176 nM for wild type KRas and various KRas mutants). Inhibits nucleotide binding to KRas in a concentration dependent manner. Displays cytotoxicity in KRas-driven cancer cell lines and inhibits downstream ERK-MAPK signaling. Cell permeable.

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      • SAHM1

        Ref: TP2117
        Sizes: 1 mg
        From: DKK8,333.00

        SAHM1 (Legacy Tebubio ref. 282TP2117). Notch pathway inhibitor - stabilized hydrocarbon-stapled alpha helical peptide. Targets the protein-protein interface and prevents Notch complex assembly.

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