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Chemicals & Small Molecules

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    Results for Chemicals & Small Molecules ( 97553 )

      • AMY-101 TFA

        Ref: TP2139L
        Sizes: 2 mg
        From: DKK4,890.00

        AMY-101 TFA (Legacy Tebubio ref. 282TP2139L). AMY-101 TFA (Cp40 TFA) is a peptidic inhibitor of the central complement component C3 (KD: 0.5 nM). AMY-101 TFA shows a favorable anti-inflammatory activity in models with COVID-19 severe pneumonia with systemic hyper inflammation.

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      • Balixafortide TFA (1051366-32-5 free base)

        Ref: TP2141
        Sizes: 5 mg, 25 mg, 50 mg
        Price Enquiry

        Balixafortide TFA (1051366-32-5 free base) (Legacy Tebubio ref. 282TP2141). Balixafortide TFA (POL6326 TFA) is a selective, well-tolerated peptidic CXCR4 antagonist (IC50 < 10 nM). It shows 1000-fold selective for CXCR4 than a large panel of receptors including CXCR7. Balixafortide TFA blocks β-arrestin recruitment and calcium flux (IC50s < 10 nM).

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      • LSKL TFA

        Ref: TP2147
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: DKK330.00

        LSKL TFA (Legacy Tebubio ref. 282TP2147). LSKL TFA (H-Leu-Ser-Lys-Leu-NH2 TFA) is a LAP-TGFβ derivative and a TGF-β1 antagonist that can cross the blood-brain barrier, inhibits the binding of TSP-1 to LAP and reduces renal interstitial fibrosis and liver fibrosis, inhibits subarachnoid fibrosis by inhibiting TSP-1-mediated TGF-β1 activity, prevents the occurrence of chronic hydrocephalus and improves long-term neurocognitive deficits after subarachnoid hemorrhage.

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      • Ramoplanin

        Ref: TP2152
        Sizes: 5 mg, 10 mg, 2 mg
        From: DKK390.00

        Ramoplanin (Legacy Tebubio ref. 282TP2152). Ramoplanin is an antibiotic extracted from Actinoplanes spp., a topical lipoglycopeptide antibacterial agent that inhibits gram-positive bacteria by binding to a critical lipid II intermediate, preventing peptidoglycan formation in the cell wall.

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      • Substance P TFA

        Ref: TP2155
        Sizes: 1 mg, 5 mg, 25 mg, 10 mg
        From: DKK405.00

        Substance P TFA (Legacy Tebubio ref. 282TP2155). Substance P TFA (Neurokinin P TFA) is a neuropeptide that functions as both a neurotransmitter and neuromodulator in the central nervous system, specifically targeting the neurokinin 1 receptor (NK1-receptor, NK1R).

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      • TRV-120027 TFA

        Ref: TP2158
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: DKK330.00

        TRV-120027 TFA (Legacy Tebubio ref. 282TP2158). TRV-120027 TFA is an angiotensin II–mediated vasoconstriction inhibitor and increases cardiomyocyte contractility. TRV-120027 TFA is a β-arrestin-1-biased AT1R agonist engaging ß-arrestins while blocking G-protein signaling[1]. TRV-120027 TFA induces acute catecholamine secretion through cation channel subfamily C3 (TRPC3) coupling and promotes the formation of a macromolecular complex composed of AT1R–β-arrestin-1–TRPC3–PLCγ at the plasma membrane.

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      • TRV-120027 acetate (1234510-46-3 free base)

        Ref: TP2158L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg
        From: DKK855.00

        TRV-120027 acetate (1234510-46-3 free base) (Legacy Tebubio ref. 282TP2158L1). TRV-120027 acetate is a β-arrestin-1-biased agonist of the angiotensin II receptor type 1 (AT1 receptor) and engages -arrestins while blocking G-protein signaling.

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      • YAP-TEAD-IN-1 TFA

        Ref: TP2160L
        Sizes: 1 mg, 5 mg, 10 mg
        From: DKK1,283.00

        YAP-TEAD-IN-1 TFA (Legacy Tebubio ref. 282TP2160L). YAP-TEAD-IN-1 TFA, a competitive inhibitor of the YAP–TEAD interaction (IC50: 25 nM), exhibits higher binding affinity to TEAD1 (Kd: 15 nM) compared to YAP (50-171) (Kd: 40 nM).

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      • YAP-TEAD-IN-1 acetate

        Ref: TP2160L1
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg
        From: DKK1,253.00

        YAP-TEAD-IN-1 acetate (Legacy Tebubio ref. 282TP2160L1). YAP-TEAD-IN-1 acetate is an effective and competitive inhibitor of YAP–TEAD interaction with an IC50 of 25 nM.

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