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Chemicals & Small Molecules

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    Results for Chemicals & Small Molecules ( 97557 )

      • GSK180

        Ref: T15426
        Sizes: 5 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: DKK735.00

        GSK180 (Legacy Tebubio ref. 282T15426). GSK180 is a selective competitive inhibitor of kynurenine 3-monooxygenase (KMO; IC50: ~6 nM), an enzyme involved in tryptophan metabolism.

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      • GSK2033

        Ref: T15427
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg
        From: DKK375.00

        GSK2033 (Legacy Tebubio ref. 282T15427). GSK2033 is an antagonist of LXR (pIC50s: 7 and 7.4 for LXRα or LXRβ, respectively).

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      • Uprosertib hydrochloride

        Ref: T15428
        Sizes: 25 mg, 100 mg, 50 mg
        From: DKK23,160.00

        Uprosertib hydrochloride (Legacy Tebubio ref. 282T15428). Uprosertib hydrochloride is a potent and selective inhibitor of pan-Akt (IC50: 180/328/38 nM for Akt1/Akt2/Akt3, respectively).

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      • GSK2194069

        Ref: T15429
        Sizes: 2 mg
        From: DKK1,275.00

        GSK2194069 (Legacy Tebubio ref. 282T15429). GSK2194069 is an active β-keto reductase (KR)-specific inhibitor of fatty acid synthase (FASN) with an IC50 of 7.7 nM in an assay for the detection of released CoA.GSK2194069 inhibits the proliferation of FAS in cancer cells through the action of acetoacetyl-coenzyme A and NADPH.

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      • Naftifine hydrochloride

        Ref: T1543
        Sizes: 1 g, 100 mg, 500 mg, 1 mL * 10 mM (in DMSO)
        From: DKK263.00

        Naftifine hydrochloride (Legacy Tebubio ref. 282T1543). Naftifine Hydrochloride is the hydrochloride salt form of naftifine, an allylamine derivate with synthetic broad-spectrum antifungal activity. Although the exact mechanism through which naftifine hydrochloride exerts its effect is unknown, it appears to selectively inhibit the enzyme squalene 2, 3-epoxidase, thereby inhibiting the biosynthesis of sterol. This results in a decreased amount of sterols, especially ergosterol which is the primary fungal membrane sterol, and a corresponding accumulation of squalene in fungal cells. Naftifine hydrochloride (Naftifine HCl) can be fungicidal as well as fungistatic to yeasts depending on the concentration and the organisms involved.

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      • GSK2256294A

        Ref: T15430
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg
        From: DKK833.00

        GSK2256294A (Legacy Tebubio ref. 282T15430). GSK2256294A (GSK 2256294) is potent, selective inhibitor of recombinant human, rat and mouse sEH with IC50 of 27 pM, 61 pM and 189 pM, respectively.

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      • Nemiralisib

        Ref: T15431
        Sizes: 1 mg, 5 mg, 25 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: DKK345.00

        Nemiralisib (Legacy Tebubio ref. 282T15431). Nemiralisib（GSK-2269557 free base） is an orally available, potent and specific PI3Kδ inhibitor with a pKi of 9.9.Nemiralisib is used for the treatment of respiratory diseases including chronic obstructive pulmonary disease.

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      • GSK256073

        Ref: T15432
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: DKK578.00

        GSK256073 (Legacy Tebubio ref. 282T15432). GSK256073 is an orally active GPR109A agonist. GSK256073 also is a long-lasting and non-flushing HCA2 (hydroxy-carboxylic acid receptor 2) full agonist (pEC50: 7.5). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis.

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      • GSK2795039

        Ref: T15433
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: DKK578.00

        GSK2795039 (Legacy Tebubio ref. 282T15433). GSK2795039 inhibits reactive oxygen species (ROS) production and NADPH consumption. GSK2795039 decreases apoptosis. GSK2795039 is an inhibitor of NADPH oxidase 2 (NOX2) (pIC50: 6 in different cell-free assays).

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