Skip to main content
Customer Service: +45 42 72 02 70
Contact us
(0)
My Wishlist
(0)
My Wishlist
(0)
My WishlistContact us
Products banner

Chemicals & Small Molecules

Filters

    Results for Chemicals & Small Molecules ( 97587 )

      • AG-370

        Ref: T21784
        Sizes: 1 mg, 5 mg, 25 mg, 10 mg
        From: DKK1,223.00

        AG-370 (Legacy Tebubio ref. 282T21784). AG 370, an indole tyrphostin, is a potent inhibitor of PDGF-induced mitogenesis with an IC50 of 20 μM, and it shows weak inhibition of the EGF receptor.

        Product detail

      • AG957

        Ref: T21785
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: DKK780.00

        AG957 (Legacy Tebubio ref. 282T21785). Tyrphostin AG957, a tyrosine kinase inhibitor with anti-BCR/ABL tyrosine kinase activity restores beta1 integrin-mediated adhesion and inhibitory signaling in chronic myelogenous leukemia hematopoietic progenitors[1].

        Product detail

      • Apogossypolone (ApoG2)

        Ref: T21786
        Sizes: 25 mg, 100 mg, 50 mg
        From: DKK12,945.00

        Apogossypolone (ApoG2) (Legacy Tebubio ref. 282T21786). Apogossypolone (ApoG2) is a semi-synthesized derivative of gossypol which is a nonpeptidic small molecule inhibitor targeting Bcl-2 family proteins with K i values of 35, 25 and 660 nM for Bcl-2, Mcl-1 and Bcl-X L, respectively. Apogossypolone shows antitumor activities, induces cell apoptosis [1] and autophagy [2]. Apogossypolone also has antifungal activity [3].

        Product detail

      • B-HT 933 dihydrochloride

        Ref: T21787
        Sizes: 1 mg, 5 mg, 10 mg
        From: DKK668.00

        B-HT 933 dihydrochloride (Legacy Tebubio ref. 282T21787). Azepexole dihydrochloride (B-HT 933), a potent and selective alpha 2-adrenoceptor agonist, exhibits affinity for α2A-, α2B-, and α2C-adrenoceptor subtypes with pKis of 8.3, 7.6, and 7.5, respectively [1]. It elicits a concentration-dependent inhibition of peristaltic contractions, evidenced by an IC50 of 78.72 nM.

        Product detail

      • Azepexole hydrochloride

        Ref: T21787L
        Sizes: 5 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: DKK263.00

        Azepexole hydrochloride (Legacy Tebubio ref. 282T21787L). Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic effects.

        Product detail

      • BD 1008 dihydrobromide

        Ref: T21788
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: DKK503.00

        BD 1008 dihydrobromide (Legacy Tebubio ref. 282T21788). BD 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors.

        Product detail

      • Triptolide

        Ref: T2179
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: DKK315.00

        Triptolide (Legacy Tebubio ref. 282T2179). Triptolide (PG490) belongs to the tricyclic diterpenoid group of natural products and is an inhibitor of NF-κB activation. Triptolide exhibits immunosuppressive, anti-rheumatic, anti-inflammatory, anti-proliferative and anti-tumor activities.

        Product detail

      • BMS 182874 hydrochloride

        Ref: T21790
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: DKK630.00

        BMS 182874 hydrochloride (Legacy Tebubio ref. 282T21790). BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.

        Product detail

      • CGP 3466B maleate

        Ref: T21792
        Sizes: 2 mg, 1 mL * 10 mM (in DMSO)
        From: DKK263.00

        CGP 3466B maleate (Legacy Tebubio ref. 282T21792). CGP 3466B maleate (Omigapil maleate) is an orally bioavailable GAPDH nitrosylation inhibitor. Omigapil maleate abrogates Aβ1-42-induced tau acetylation, memory impairment, and locomotor dysfunction in mice. Omigapil maleate has the potential for the research of Alzheimer's disease. Omigapil maleate (CGP3446B maleate) is a apoptosis inhibitor. Omigapil maleate can be used for the research of congenital muscular dystrophy (CMD).

        Product detail