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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70877 )

      • AMN082

        Ref: T21935
        Sizes: 1 mg, 5 mg, 25 mg, 10 mg

        AMN082 (Legacy Tebubio ref. 282T21935). AMN082 is an mGluR7 agonist with antidepressant effects. AMN082 has a neuroprotective effect on neuronal apoptosis in rats with traumatic brain injury and attenuates cocaine- and morphine-induced locomotor sensitization and cross-sensitization in mice.

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      • AMN082 free base

        Ref: T21935L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg

        AMN082 free base (Legacy Tebubio ref. 282T21935L). AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.

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      • M50054

        Ref: T21936
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)

        M50054 (Legacy Tebubio ref. 282T21936). Apoptosis Inhibitor was a novel inhibitor of programmed cell death associate with caspase-3 inhibition.

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      • AS-041164

        Ref: T21938
        Sizes: 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)

        AS-041164 (Legacy Tebubio ref. 282T21938). AS-041164 is a selective and orally active PI3Kγ isoform inhibitor(IC50 of 70 nM), and shows less activity against PI3Kα, PI3Kβ, and PI3Kδ (IC50s of 240 nM, 1.45 μM, and 1.70 μM, respectively). It has anti-inflammatory effects.

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      • ATB-337

        Ref: T21939
        Sizes: 1 mg, 5 mg, 50 mg, 10 mg

        ATB-337 (Legacy Tebubio ref. 282T21939). S-Diclofenac is a novel NSAID formed by linking diclofenac to an H2S-releasing moiety. S-Diclofenac spares the gastric mucosa of injury despite markedly suppressing prostaglandin synthesis [1].

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      • Direct Blue 1

        Ref: T2194
        Sizes: 500 mg, 1 mL * 10 mM (in DMSO)

        Direct Blue 1 (Legacy Tebubio ref. 282T2194). Direct Blue 1 (Pontamine sky blue), a counterstain for background autofluorescence in immunofluorescence histochemistry, structurally resembles glutamate and operates as a potent, competitive VGLUT inhibitor, not impacting plasma membrane transporters. This compound stands out as the inaugural small molecule PrP ligand to inhibit Aβ binding.

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      • BIM 23056 Acetate

        Ref: T21944L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)

        BIM 23056 Acetate (Legacy Tebubio ref. 282T21944L). BIM 23056 Acetate is a  potent and surmountable human recombinant sst5 receptor antagonist.

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      • BIMU 8

        Ref: T21946
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)

        BIMU 8 (Legacy Tebubio ref. 282T21946). BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, and 540 nM for wild-type 5HT4 receptor, T3.36A, and W6.48A mutant 5-HT4.

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      • Calpain Inhibitor XII

        Ref: T21949
        Sizes: 1 mg, 5 mg, 25 mg, 50 mg, 10 mg

        Calpain Inhibitor XII (Legacy Tebubio ref. 282T21949). Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a selective and potent inhibitor of calpain I, inhibits calpain II and cathepsin B. Calpain Inhibitor XII shows antiviral activity against coronavirus in cell culture.

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