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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70877 )

      • K 00546

        Ref: T21950
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 1 mL * 10 mM (in DMSO)

        K 00546 (Legacy Tebubio ref. 282T21950). K 00546 is a potent inhibitor of cellular cyclin kinases (CDK1 and CDK2) and CDC2-like kinases (CLK1 and CLK3) used in the study of cancer and immune-related diseases.

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      • CDP 840 hydrochloride

        Ref: T21951
        Sizes: 25 mg, 100 mg, 50 mg

        CDP 840 hydrochloride (Legacy Tebubio ref. 282T21951). CDP-840 (GR259653X) is a potent, selective, and orally active phosphodiesterase IV (PDE IV) inhibitor that specifically inhibits antigen-induced early and late phase bronchoconstriction in conscious squirrel monkeys [1].

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      • EGFR/ErbB-2/ErbB-4 inhibitor-2

        Ref: T21954
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 2 mg, 1 mL * 10 mM (in DMSO)

        EGFR/ErbB-2/ErbB-4 inhibitor-2 (Legacy Tebubio ref. 282T21954). EGFR/ErbB-2/ErbB-4 inhibitor-2 (EGFR/ErbB2 Inhibitor) is a cell-permeable compound that inhibits EGFR and c-ErbB2 with IC50 values of 20 nM and 79 nM, respectively.

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      • GQ-16

        Ref: T21955
        Sizes: 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 200 mg

        GQ-16 (Legacy Tebubio ref. 282T21955). GQ-16 is a partial agonist of PPARγ with a Ki of 160 nM. GQ-16 reduces adipogenic actions and promotes insulin Sensitization without weight gain.

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      • GSK3β inhibitor II

        Ref: T21956
        Sizes: 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)

        GSK3β inhibitor II (Legacy Tebubio ref. 282T21956). GSK3β inhibitor II is a GSK3β inhibitor. GSK3β inhibitor II exhibits the research potential of Alzheimer's disease (AD).

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      • Guanabenz hydrochloride

        Ref: T21957
        Sizes: 100 mg, 50 mg, 500 mg, 200 mg, 1 mL * 10 mM (in DMSO)

        Guanabenz hydrochloride (Legacy Tebubio ref. 282T21957). Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.

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      • Fipronil

        Ref: T2196
        Sizes: 1 g, 100 mg, 50 mg, 500 mg, 200 mg, 1 mL * 10 mM (in DMSO)

        Fipronil (Legacy Tebubio ref. 282T2196). Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family. Fipronil is a broad-spectrum insecticide that disrupts the insect central nervous system by blocking GABA-gated chloride channels and glutamate-gated chloride (GluCl) channels, resulting in central nervous system toxicity. This causes hyperexcitation of contaminated insects' nerves and muscles. Specificity of fipronil on insects may come from a better efficacy on GABA receptor, but also because GluCl channels do not exist in mammals.

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      • HZ52

        Ref: T21962
        Sizes: 1 mg, 5 mg, 25 mg, 10 mg

        HZ52 (Legacy Tebubio ref. 282T21962). HZ52 is a potent, reversible 5-lipoxygenase (5-LO) inhibitor that blocks leukotriene (LTs) synthesis with an IC50 of 0.7 μM in intact human polymorphonuclear leukocytes [1].

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      • MBCQ

        Ref: T21965
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)

        MBCQ (Legacy Tebubio ref. 282T21965). MBCQ is an inhibitor of cGMP-specific phosphodiesterase PDE5.

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