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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70877 )

      • P32/98 hemifumarate

        Ref: T21979
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg

        P32/98 hemifumarate (Legacy Tebubio ref. 282T21979). P32/98 hemifumarate is a dipeptidyl peptidase IV (DPP4) inhibitor with hypoglycemic properties that improves insulin sensitivity and β-cell responsiveness in the Zucker diabetic rat model, and may be useful in studies of type 2 diabetes and colitis.

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      • Arecoline hydrobromide

        Ref: T2198
        Sizes: 50 mg, 1 mL * 10 mM (in DMSO)

        Arecoline hydrobromide (Legacy Tebubio ref. 282T2198). Arecoline hydrobromide (Arecoline HBr) is a muscarinic acetylcholine receptor agonist.

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      • PD 198306

        Ref: T21980
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)

        PD 198306 (Legacy Tebubio ref. 282T21980). PD 198306 is a selective inhibitor of MAPK/ERK-kinase (MEK) with antihyperalgesic effects. PD 198306 reduces the Streptozocin-induced increase in the level of active ERK1.

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      • Phthalazinone pyrazole

        Ref: T21981
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 2 mg

        Phthalazinone pyrazole (Legacy Tebubio ref. 282T21981). Phthalazinone pyrazole is potent, selective, and orally bioavailable inhibitor of Aurora-A kinase. Aurora-A is overexpressed in a variety of tumor types and displays oncogenic activity.

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      • PKI 14-22 amide, myristoylated Acetate

        Ref: T21983L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)

        PKI 14-22 amide, myristoylated Acetate (Legacy Tebubio ref. 282T21983L). PKI 14-22 amide, myristoylated Acetate inhibit cAMP-dependent protein kinase (PKA) and blocks hyperalgesia produced by spinal administration of 8-bromo-cAMP. 

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      • PT-1

        Ref: T21984
        Sizes: 1 mg, 5 mg, 25 mg, 50 mg, 10 mg

        PT-1 (Legacy Tebubio ref. 282T21984). PT-1 is an AMPKα1 activator that dose-dependently activates AMPK α1394, α1335, and α2398 and enhances AMPK phosphorylation.

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      • SSR 69071

        Ref: T21989
        Sizes: 1 mg, 5 mg, 10 mg

        SSR 69071 (Legacy Tebubio ref. 282T21989). SSR69071 is a potent, orally active, and selective inhibitor of neutrophil elastase, displaying higher affinity for human elastase (Ki = 0.0168 nM) compared to rat (Ki = 3 nM), mouse (Ki = 1.8 nM), and rabbit (Ki = 58 nM) elastases [2]. It reduces myocardial infarct size following ischemia-reperfusion injury [1] and has potential for treating chronic obstructive pulmonary diseases, asthma, emphysema, cystic fibrosis, and various inflammatory diseases.

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      • Myclobutanil

        Ref: T2199
        Sizes: 100 mg, 50 mg, 500 mg, 1 mL * 10 mM (in DMSO)

        Myclobutanil (Legacy Tebubio ref. 282T2199). Myclobutanil (Systhane) is a triazole chemical used as a fungicide. It is a steroid demethylation inhibitor, specifically inhibiting ergosterol biosynthesis. Ergosterol is a critical component of fungal cell membranes.

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      • Vacuolin-1

        Ref: T21992
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg

        Vacuolin-1 (Legacy Tebubio ref. 282T21992). Vacuolin-1 is a cell-permeable inhibitor of Ca2+ dependent fusion of lysosomes to the cell membrane. It acts by inhibiting release of lysosomal content.vacuolin‐1 is a potent and selective PIKfyve inhibitor and inhibits late‐stage autophagy by impairing lysosomal maturation

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