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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70877 )

      • AGK7

        Ref: T22026
        Sizes: 1 mg, 5 mg, 25 mg, 10 mg

        AGK7 (Legacy Tebubio ref. 282T22026). AGK7 is an inactive control of AGK2, a selective SIRT2 inhibitor that selectively inhibits SIRT3 over SIRT1 and SIRT2 (IC50 = >5 μM, >50 μM and >50 μM for SIRT3, SIRT1, and SIRT2, respectively).

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      • AH-7614

        Ref: T22027
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)

        AH-7614 (Legacy Tebubio ref. 282T22027). AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist.

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      • AL 34662

        Ref: T22029
        Sizes: 1 mg, 5 mg, 25 mg, 10 mg

        AL 34662 (Legacy Tebubio ref. 282T22029). AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also a low affinity α-1D adrenergic agonist, with an EC50 of 0.4 μM.AL 34662 can be used to lower intraocular pressure.

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      • D-Carnitine hydrochloride

        Ref: T2203
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)

        D-Carnitine hydrochloride (Legacy Tebubio ref. 282T2203). D-Carnitine hydrochloride ((S)-Carnitine Hydrochloride) is a component of striated muscle and liver, used therapeutically to stimulate gastric and pancreatic secretions and to treat hyperlipoproteinemias.

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      • ANR 94

        Ref: T22031
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 2 mg, 1 mL * 10 mM (in DMSO)

        ANR 94 (Legacy Tebubio ref. 282T22031). ANR94 is a potent, selective antagonist of the adenosine A2A receptor (AA2AR), exhibiting a K_i value of 46 nM for the human AA2AR (hAA2AR). This compound shows promise for research into Parkinson's disease. [1] [2]

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      • ARC 239 dihydrochloride

        Ref: T22033
        Sizes: 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)

        ARC 239 dihydrochloride (Legacy Tebubio ref. 282T22033). ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist with pKD values of 8.8, 6.7, and 6.4 at α2B, α2A, and α2D receptors respectively (pKD values are 8.8, 6.7, and 6.4 at α2B, α2A, and α2D receptors respectively).

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      • ARP 101

        Ref: T22034
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)

        ARP 101 (Legacy Tebubio ref. 282T22034). ARP 101 is an effective selective matrix metalloproteinase-2 (MMP-2) inhibitor with anti-cancer activity. It induces the inhibition of HCMV through non-classical chelate 1 (SQSTM1)/p62-Keap1-Nrf2 pathways and phosphorylation of the C-terminal domain of p62, regulating autophagy and inhibiting melanogenesis.

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      • Arylquin 1

        Ref: T22036
        Sizes: 1 mg, 5 mg, 10 mg

        Arylquin 1 (Legacy Tebubio ref. 282T22036). Arylquin 1, a prostate-apoptosis-response-4 (Par-4) secretagogue, specifically targets vimentin to facilitate Par-4 secretion. It also induces lysosomal membrane permeabilization (LMP) and promotes non-apoptotic cell death in cancer cells [1].

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      • AS 1892802

        Ref: T22037
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)

        AS 1892802 (Legacy Tebubio ref. 282T22037). AS 1892802 is a potent and selective inhibitor of ROCK. AS 1892802 exibits IC50 values of 52nM, 57nM and 122 nM for human ROCK2, rat ROCK2 and human ROCK1, respectively. The onset of antinociceptive effect of AS 1892802 is as fast as those of Tramadol and Diclofenac.

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