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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70877 )

      • PTP Inhibitor IV

        Ref: T22137
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)

        PTP Inhibitor IV (Legacy Tebubio ref. 282T22137). PTP Inhibitor IV is an effective protein tyrosine phosphatase (PTP) inhibitor, which can selectively inhibit DUSP14 phosphatase activity (IC50.5.21μm). PTP Inhibitor IV inhibited SHP-2, PTP1B, PTp-ε, PTP Meg-2, PTP-σ, PTP-β and PTP-μ, IC50 were 1.8 μM, 2.5 μM, 8.4 μM, 13 μM, 20 μM, 6.4 μM, and 6.7 μM, respectively. PTP Inhibitor IV affects cellular signaling by inhibiting PTP activity and may regulate specific pathways associated with PTP-mediated signaling events.

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      • Flumethrin

        Ref: T2214
        Sizes: 5 mg, 25 mg, 10 mg, 2 mg

        Flumethrin (Legacy Tebubio ref. 282T2214). Flumethrin is a pyrethroid insecticide. It is used externally in veterinary medicine against parasitic insects and ticks on cattle, sheep, goats, horses, and dogs, and the treatment of parasitic mites in honeybee colonies.

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      • (R)-SLV 319

        Ref: T22140
        Sizes: 5 mg, 10 mg

        (R)-SLV 319 (Legacy Tebubio ref. 282T22140). (R)-SLV 319 is a potent and selective antagonist of cannabinoid receptor 1 (CB1) with a Ki value of 894 nM. It is the dextrorotatory counterpart of SLV 319 [1].

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      • RO8191

        Ref: T22142
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg

        RO8191 (Legacy Tebubio ref. 282T22142). RO8191 (CDM-3008) (CDM-3008) is an agonist of interferon (IFN) receptor.

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      • (S)-Lisofylline

        Ref: T22148
        Sizes: 1 mg, 1 mL * 10 mM (in DMSO)

        (S)-Lisofylline (Legacy Tebubio ref. 282T22148). (S)-Lisofylline is the inactive optical enantiomer of (R)-lisofylline which is an anti-inflammatory agent. (S)-Lisofylline is exclusively converted to pentoxifylline in human liver microsomes.

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      • Ferulic Acid

        Ref: T2215
        Sizes: 100 mg, 50 mg, 1 mL * 10 mM (in DMSO)

        Ferulic Acid (Legacy Tebubio ref. 282T2215). Ferulic Acid (Coniferic acid) is a highly abundant phenolic phytochemical and a type of organic compound found in the Ferula assafoetida L. or Ligusticum chuanxiong.It can be absorbed by the small intestine and excreted through the urine.

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      • SR 2595

        Ref: T22154
        Sizes: 1 mg, 5 mg, 10 mg

        SR 2595 (Legacy Tebubio ref. 282T22154). SR2595 is an inverse agonist of the nuclear receptor PPARγ with an IC₅₀ of 30 nM [1].

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      • TCS 2002

        Ref: T22157
        Sizes: 50 mg

        TCS 2002 (Legacy Tebubio ref. 282T22157). GSK-3β inhibitor 9 (Compound 9b) is a highly selective, orally bioavailable and potent GSK-3β inhibitor with the IC 50 of 35 nM. GSK-3β inhibitor 9 exhibits good pharmacokinetic profiles including favorable BBB penetration. GSK-3β inhibitor 9 is able to be used for the research of Alzheimer’s disease [1].

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      • TCS 3035

        Ref: T22158
        Sizes: 50 mg

        TCS 3035 (Legacy Tebubio ref. 282T22158). GPR35 agonist 4 (compound 10) demonstrates high potency as a GPR35 agonist with a pEC50 of 5.86, effective on both human and rat GPR35; mutation of arginine at position 3.36 results in loss of its agonist function on GPR35 [1].

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