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    Results for Activators & Inhibitors ( 70845 )

      • Ref: T22584
        Sizes: 25 mg, 100 mg, 50 mg

        Arecaidine but-2-ynyl ester tosylate (Legacy Tebubio ref. 282T22584). mAChR M2 agonist

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      • Arecaidine propargyl ester tosylate (Legacy Tebubio ref. 282T22585). Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.

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      • Ref: T22586
        Sizes: 5 mg, 100 mg, 50 mg, 10 mg

        Arvanil (Legacy Tebubio ref. 282T22586). Cannabinoid CB1 and vanilloid TRPV1 (VR1) agonist

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      • Ref: T22587
        Sizes: 5 mg, 25 mg, 10 mg

        AS-604850 (Legacy Tebubio ref. 282T22587). AS-604850 is a selective and ATP-competitive PI3Kγ inhibitor (IC50= 2.5 μM). It has over 30-fold selectivity for PI3Kδ and PI3Kβ, and 18-fold selectivity over PI3Kα.

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      • Ref: T22589
        Sizes: 1 mg

        Asenapine hydrochloride (Legacy Tebubio ref. 282T22589). Asenapine hydrochloride (Org 5222 hydrochloride) is a 5-hydroxytryptamine receptor, adrenergic receptor, dopamine receptor and histamine receptor antagonist with antipsychotic effects used in neurological disorders such as schizophrenia and bipolar disorder.

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      • Ref: T2259
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)

        Silmitasertib (Legacy Tebubio ref. 282T2259). Silmitasertib (CX-4945) is a potent, orally bioavailable inhibitor of casein kinase 2 (CK2; Ki: 0.38 nM).

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      • Ref: T22590
        Sizes: 2 mg

        AT7519 TFA (Legacy Tebubio ref. 282T22590). AT7519 is a kinase inhibitor (IC50: 0.19, 0.044, 0.51, 0.067, 0.66 and 0.018 μM for CDK1/cyclinB, CDK2/CyclinA, CDK2/Cyclin E, CDk4/CyclinD1, CDK6/Cyclin D3, CDk5/p35).

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      • Ref: T22591
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg

        ATC 0175 hydrochloride (Legacy Tebubio ref. 282T22591). ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective. ATC 0175 hydrochloride has affinity for MCH1R, MCH2R, MCH1, 5-HT2B receptors and 5-HT1A receptors with IC50s of 13.5 nM, >10,000 nM, 13 nM, 9.66 nM and 16.9 nM, respectively. ATC 0175 hydrochloride exhibits antidepressant and anxiolytic effects in animal models. aTC 0175 can be used to study depression and/or anxiety disorders.

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      • Ref: T22592
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg

        ATPγS tetralithium salt (Legacy Tebubio ref. 282T22592). ATPγS tetralithium salt is a good substrate for RNA-stimulated nucleotide hydrolysis and RNA unwinding activity of eIF4A.

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