Skip to main content
Customer Service: +45 42 72 02 70
Contact us
(0)
My Wishlist
(0)
My Wishlist
(0)
My WishlistContact us
Products banner

Activators & Inhibitors

Filters

    Results for Activators & Inhibitors ( 70846 )

      • CS 2100

        Ref: T22697
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg

        CS 2100 (Legacy Tebubio ref. 282T22697). CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.

        Product detail

      • TLR3-IN-1

        Ref: T22698
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)

        TLR3-IN-1 (Legacy Tebubio ref. 282T22698). TLR3-IN-1 (CU CPT 4a) is a selective TLR3 inhibitor (IC50: 3.44 μM in RAW 264.7 cells). It can inhibit TLR3/dsRNA complex-mediated downstream signaling pathways and inhibit the production of TNF-α and IL-1β in whole cells.

        Product detail

      • Cyanopindolol hemifumarate

        Ref: T22699
        Sizes: 25 mg, 100 mg, 50 mg

        Cyanopindolol hemifumarate (Legacy Tebubio ref. 282T22699). 5-HT1A/1B antagonist and β-adrenoceptor antagonist

        Product detail

      • Trans-Tranilast

        Ref: T2270
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)

        Trans-Tranilast (Legacy Tebubio ref. 282T2270). Trans-Tranilast is an antiallergic drug developed by Kissei Pharmaceuticals. It was approved in 1982 for use in Japan and South Korea for bronchial asthma. Indications for keloid and hypertrophic scar were added in 1993. It has been used for the treatment of allergic disorders such as asthma, allergic rhinitis and atopic dermatitis.

        Product detail

      • Cyclapolin 9

        Ref: T22700
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)

        Cyclapolin 9 (Legacy Tebubio ref. 282T22700). Cyclapolin 9 is a selective, potent, and ATP-competitive inhibitor of polo-like kinase 1 (PLK1) with an IC50 of 500 nM, and has not shown activity against other kinases.

        Product detail

      • CYM 50769

        Ref: T22702
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg

        CYM 50769 (Legacy Tebubio ref. 282T22702). CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM). CYM 50769 inhibited NPW activation of NPBWR1 with a submicromolar IC50, and displayed high selectivity against a broad array of off-targets with pharmaceutical relevance.

        Product detail

      • CYM-5520

        Ref: T22703
        Sizes: 1 mg, 100 mg, 10 mg

        CYM-5520 (Legacy Tebubio ref. 282T22703). CYM-5520 is a noncompetitive allosteric agonist of S1P2

        Product detail