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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70846 )

      • ONO-2952

        Ref: T16393
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,896.00

        ONO-2952 (Legacy Tebubio ref. 282T16393). ONO-2952 is more selective for TSPO than other receptors, transporters, ion channels, and enzymes. ONO-2952 is a potent and selective translocator protein 18 kDa (TSPO) antagonist (Ki: 0.33-9.30 nM for rat and human TSPO). ONO-2952 has the potential for irritable bowel syndrome treatment. ONO-2952 exerts its anti-stress effects through inhibition of excessive activation of the noradrenergic system in the brain without the amnesic effect.

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      • ONO-5334

        Ref: T16394
        Sizes: 1 mg, 5 mg, 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €188.00

        ONO-5334 (Legacy Tebubio ref. 282T16394). ONO-5334 is a selective, orally active and potent histone K inhibitor with anti-SAR-COV-2 and anti-bone resorption activity for the study of osteoporosis.

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      • ONO4057

        Ref: T16395
        Sizes: 1 mg, 5 mg
        From: €795.00

        ONO4057 (Legacy Tebubio ref. 282T16395). ONO4057 is a potent and orally active Leukotriene B4 receptor antagonist with an IC50 value of 0.7±0.3 μM. Immunosuppressive effect of ONO4057 on rat allografts.

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      • OP-3633

        Ref: T16396
        Sizes: 25 mg
        Price Enquiry

        OP-3633 (Legacy Tebubio ref. 282T16396). OP-3633 is an effective and selective steroidal glucocorticoid receptor (GR) antagonist (IC50: 29 nM). OP-3633 shows low progesterone receptor (PR) agonism and androgen receptor (AR) antagonism. It also has an inhibition of GR transcriptional activity.

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      • Ophiobolin A

        Ref: T16397
        Sizes: 1 mg
        From: €781.00

        Ophiobolin A (Legacy Tebubio ref. 282T16397). Ophiobolin A is a fungal metabolite and a phytotoxin and is an effective and irreversibly inhibitor of calmodulin-activated cyclic nucleotide phosphodiesterase (IC50: 9 μM). Ophiobolin A also has antimicrobial and anticancer activity.

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      • Opicapone

        Ref: T16398
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €67.00

        Opicapone (Legacy Tebubio ref. 282T16398). Opicapone (BIA 9-1067) reduces the ATP content of the cells (IC50: 98 μM). Opicapone is an effective third-generation catechol-O-methyltransferase inhibitor for the research of Parkinson's disease and motor fluctuations.

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      • Opiranserin

        Ref: T16399
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        Opiranserin (Legacy Tebubio ref. 282T16399). Opiranserin is a development as an injectable agent for the treatment of postoperative pain. Opiranserin is a non-opioid and non-NSAID analgesic candidate and is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A) (IC50s: 0.86 and 1.3 μM, respectively). Opiranserin displays antagonistic activity on rP2X3 (IC50=0.87 μM).

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      • Ciprofloxacin

        Ref: T1640
        Sizes: 1 g, 500 mg
        From: €47.00

        Ciprofloxacin (Legacy Tebubio ref. 282T1640). Ciprofloxacin (Bay-09867), a synthetic broad spectrum fluoroquinolone antibiotic, inhibits bacterial DNA gyrase. It is more active against Gram-negative bacteria than Gram-positive bacteria.

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      • Org-12962

        Ref: T16401
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €46.00

        Org-12962 (Legacy Tebubio ref. 282T16401). Org-12962 is an effective and selective 5-HT2C receptor agonist pEC50: 7.01). Org-12962 shows antiaversive effects in a rat model of panic-like anxiety. Org-12962 also shows high effacy for the 5-HT2A and 5-HT2B receptors (pEC50s: 6.38 and 6.28, respectively).

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