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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70847 )

      • Lenalidomide

        Ref: T1642
        Sizes: 1 g, 100 mg, 50 mg, 500 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €41.00

        Lenalidomide (Legacy Tebubio ref. 282T1642). Lenalidomide (CC-5013) is an immunomodulator with oral activity. Lenalidomide is a ligand for the ubiquitin E3 ligase cereblon (CRBN), which selectively ubiquitinates and degrades two lymphoid transcription factors, IKZF1 and IKZF3, via the CRBN-CRL4 ubiquitin ligase, and is commonly used in the synthesis of PROTAC products.

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      • P-1075

        Ref: T16420
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €63.00

        P-1075 (Legacy Tebubio ref. 282T16420). P-1075 is a potent sulfonylurea receptor 2-associated ATP-sensitive potassium channels (SUR2-KIR6) activator (EC50 = 45 nM). P-1075 opens opens mitoKATP channels and may be cardioprotective.

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      • p-MPPI hydrochloride

        Ref: T16421
        Sizes: 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €97.00

        p-MPPI hydrochloride (Legacy Tebubio ref. 282T16421). p-MPPI hydrochloride is a selective 5-HT1A receptor antagonist with antidepressant and anxiolytic-like effects.

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      • P110δ-IN-1

        Ref: T16422
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: €46.00

        P110δ-IN-1 (Legacy Tebubio ref. 282T16422). P110δ-IN-1 (PWT-143) is an effective and selective inhibitor of P110δ (IC50: 8.4 nM).

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      • p32 Inhibitor M36

        Ref: T16423
        Sizes: 100 mg, 2 mg
        From: €102.00

        p32 Inhibitor M36 (Legacy Tebubio ref. 282T16423). p32 inhibitor M36 is an inhibitor of p32 mitochondrial protein. It binds directly to p32 and inhibits the p32 association with LyP-1.

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      • p38 MAPK-IN-1

        Ref: T16424
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €225.00

        p38 MAPK-IN-1 (Legacy Tebubio ref. 282T16424). p38 MAPK-IN-1 displays sustained levels, low clearance, and good bioavailability. p38 MAPK-IN-1 is a novel effective and selective inhibitor of p38 MAPK (IC50: 68 nM).

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      • PA452

        Ref: T16425
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €96.00

        PA452 (Legacy Tebubio ref. 282T16425). PA452 is a selective antagonist of retinoic X receptor (RXR) and suppresses the effect of Retinoic acid on Th1/Th2 development.

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      • Asivatrep

        Ref: T16426
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 1 mL * 10 mM (in DMSO)
        From: €394.00

        Asivatrep (Legacy Tebubio ref. 282T16426). Asivatrep (PAC14028) is a selective and potent antagonist of transient receptor potential vanilloid subtype 1 (TRPV1) for the study of atopic dermatitis.

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      • Padsevonil

        Ref: T16427
        Sizes: 1 mg
        From: €283.00

        Padsevonil (Legacy Tebubio ref. 282T16427). Padsevonil (UCB-0942) is a potential GABA A receptor orthosteric modulator with antiepileptic activity for the treatment of epilepsy.

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