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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70847 )

      • Pafuramidine

        Ref: T16428
        Sizes: 1 mg, 5 mg, 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €112.00

        Pafuramidine (Legacy Tebubio ref. 282T16428). Pafuramidine (DB289) is an experimental prodrug of the orally active metabolite DB75, a potent antiparasitic compound with anti-malarial activity used in the study of parasitic infections and sleeping sickness.

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      • GNE 2861

        Ref: T16429
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €41.00

        GNE 2861 (Legacy Tebubio ref. 282T16429). GNE 2861 inhibits PAK4, PAK5, and PAK6 (IC50s: 7.5, 36, 126 nM, respectively). GNE 2861 is a PAK inhibitor that shows group II selectivity.

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      • Penciclovir

        Ref: T1643
        Sizes: 100 mg, 500 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €33.00

        Penciclovir (Legacy Tebubio ref. 282T1643). Penciclovir (BRL 39123) is a Herpesvirus Nucleoside Analog DNA Polymerase Inhibitor. In HSV infected cells, penciclovir is phosphorylated by viral thymidine kinase and subsequently converted by cellular kinases into the active metabolite, penciclovir triphosphate, which competitively inhibits viral HSV polymerase by blocking deoxyguanosine triphosphate substrate binding. As a result, herpes viral DNA synthesis and replication are selectively inhibited.

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      • Paliroden

        Ref: T16430
        Sizes: 1 mg, 5 mg
        From: €795.00

        Paliroden (Legacy Tebubio ref. 282T16430). Paliroden is a non-peptide compound that can be taken orally and is used for supplementing neuro-nutrition. It stimulates the synthesis of endogenous neurotrophic factors and is employed in the research of neurodegenerative diseases such as Alzheimer's and Parkinson's.

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      • Pamatolol

        Ref: T16431
        Sizes: 1 mg, 5 mg
        From: €795.00

        Pamatolol (Legacy Tebubio ref. 282T16431). Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.

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      • Pan-RAS-IN-1

        Ref: T16432
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €83.00

        Pan-RAS-IN-1 (Legacy Tebubio ref. 282T16432). Pan-RAS-IN-1 is an inhibitor of pan-Ras. It disrupts the interaction of Ras proteins and their effectors.

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      • Pancopride

        Ref: T16433
        Sizes: 1 mg, 5 mg
        From: €795.00

        Pancopride (Legacy Tebubio ref. 282T16433). Pancopride（LAS 30451） is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-induced vomiting.

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      • PAT-048

        Ref: T16434
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,896.00

        PAT-048 (Legacy Tebubio ref. 282T16434). PAT-048 is an effective and selective autotaxin inhibitor. PAT-048 reduces dermal fibrosis in vivo. PAT-048 also inhibits IL-6 mRNA expression but displays no effect on autotaxin protein and pulmonary lysophosphatidic acid (LPA) production in the lung fibrosis model. PAT-048 has an IC50 and IC90 of 20 nM and 200 nM for autotaxin in mouse plasma.

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      • PBIT

        Ref: T16435
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €39.00

        PBIT (Legacy Tebubio ref. 282T16435). PBIT inhibits JARID1B histone demethylase (IC50 of about 3 μM). PBIT also inhibits JARID1A and JARID1C (IC50s of 6 μM and 4.9 μM, respectively). PBIT is a specific inhibitor of the Jumonji AT-rich Interactive Domain 1 (JARID1) enzymes .

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