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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70847 )

      • PF-06465469

        Ref: T16493
        Sizes: 100 mg, 50 mg
        From: €814.00

        PF-06465469 (Legacy Tebubio ref. 282T16493). PF-06465469 is a covalent ITK inhibitor(IC50: 2 nM).

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      • PF-06471553

        Ref: T16494
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,646.00

        PF-06471553 (Legacy Tebubio ref. 282T16494). PF-06471553 is an effective and selective inhibitor of monoacylglycerol acyltransferase 3 (IC50: 92 nM).

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      • PF-06795071

        Ref: T16496
        Sizes: 25 mg, 100 mg, 50 mg
        From: €2,747.00

        PF-06795071 (Legacy Tebubio ref. 282T16496). PF-06795071 is an effective and selective covalent inhibitor of MAGL (IC50: 3 nM).

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      • PF 1022A

        Ref: T16497
        Sizes: 1 mg, 5 mg
        From: €336.00

        PF 1022A (Legacy Tebubio ref. 282T16497). PF 1022A is an N-methylated cyclooctadepsipeptides with strong anthelmintic properties. It also acts as an ionosphere.

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      • Mardepodect

        Ref: T16499
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €41.00

        Mardepodect (Legacy Tebubio ref. 282T16499). Mardepodect (PF-2545920) is a phosphodiesterase inhibitor selective for the PDE10A subtype with an IC50 of 0.37 nM and over 1000-fold selectivity over PDE. It is potentially useful for the treatment of schizophrenia. Phosphodiesterase 10A (PDE10A) is highly expressed in striatal medium spiny neurons of both the direct and indirect output pathways. Mardepodect can cross the blood-brain barrier.

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      • Tenofovir hydrate

        Ref: T1649L
        Sizes: 5 mg, 25 mg, 50 mg, 10 mg
        From: €45.00

        Tenofovir hydrate (Legacy Tebubio ref. 282T1649L). Tenofovir hydrate (GS 1278 hydrate) is a nucleotide reverse transcriptase inhibitor with antiviral activity, inhibits EBV replication, and is used in the study of HIV and HBV.

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      • Chlorzoxazone

        Ref: T1650
        Sizes: 1 g, 10 g, 5 g
        From: €35.00

        Chlorzoxazone (Legacy Tebubio ref. 282T1650). Chlorzoxazone (Chlorzoxazon) is a Muscle Relaxant. The physiologic effect of chlorzoxazone is by means of Centrally-mediated Muscle Relaxation.

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      • PF-3450074

        Ref: T16500
        Sizes: 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €33.00

        PF-3450074 (Legacy Tebubio ref. 282T16500). PF-3450074 (PF-74) acts at an early stage of HIV-1 infection inhibits viral replication by directly competing with the binding of CPSF6 (nuclear host factors cleavage and polyadenylation specific factor 6) and NUP153 (nucleoporin 153), and blocks the uncoating, assembly, and the reverse transcription steps of the viral life cycle. PF-3450074 is a specifical inhibitor of HIV-1 capsid protein (CA) and shows a broad-spectrum inhibition of HIV isolates with submicromolar potency (EC50=8-640 nM).

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      • PF-3644022

        Ref: T16501
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €36.00

        PF-3644022 (Legacy Tebubio ref. 282T16501). PF-3644022 is an effective, selective, and ATP-competitive MAPKAPK2 (MK2) inhibitor (IC50: 5.2 nM and a Ki of 3 nM). PF-3644022 potently inhibits TNFα production and has an anti-inflammatory effect. PF-3644022 also inhibits MK3 and p38 regulated/activated kinase (PRAK) (IC50s: 53 nM and 5.0 nM, respectively).

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