Skip to main content
Customer Service: +31 072-572 21 00
Contact us
(0)
My Wishlist
(0)
My Wishlist
(0)
My WishlistContact us
Products banner

Activators & Inhibitors

Filters

    Results for Activators & Inhibitors ( 70846 )

      • Polyoxyethylene stearate

        Ref: T16561
        Sizes: 10 g, 5 g
        From: €52.00

        Polyoxyethylene stearate (Legacy Tebubio ref. 282T16561). Polyoxyethylene stearate (POES) is an agent of non-ionic emulsifying.

        Product detail

      • Ponceau 4R

        Ref: T16562
        Sizes: 1 g
        From: €57.00

        Ponceau 4R (Legacy Tebubio ref. 282T16562). Ponceau 4R (Acid Red 18) is a synthetic strawberry red azo dye that is a food colorant dye used in a variety of food products. It is stable to light, heat and acid, but fades in the presence of ascorbic acid. It is usually synthesized from aromatic hydrocarbons.

        Product detail

      • Pozanicline

        Ref: T16563
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        Pozanicline (Legacy Tebubio ref. 282T16563). Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction. Pozanicline selectively activate neuronal nicotinic acetylcholine receptor (nAChR) subtypes, is a novel cholinergic agent that is a partial agonist at α4β2 nAChRs (Ki=16 nM). It shows high selectivity for α6β2 and α4α5β2 nAChR subtypes, the binding affinity (Ki, rat) for Pozanicline to [3H] cytisine sites is 16.7 nM .

        Product detail

      • Pozanicline hydrochloride

        Ref: T16563L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €80.00

        Pozanicline hydrochloride (Legacy Tebubio ref. 282T16563L). Pozanicline hydrochloride is an orally bioavailable nicotinic acetylcholine receptor (nAChR) agonist with a Ki of 16.7 nM for binding to [3H]cytisine sites[1]. Pozanicline hydrochloride is an α4β2-selective nAChR agonist, which binds to rat brain α4β2 nAChR with a Ki of 17 nM while binding to α7 nAChR is insignificant[2].

        Product detail

      • PPADS tetrasodium

        Ref: T16564
        Sizes: 1 mg
        From: €50.00

        PPADS tetrasodium (Legacy Tebubio ref. 282T16564). PPADS tetrasodiuma is a potent P2X receptor antagonist and inhibitor of the inverse mode of Na/Ca²⁺ exchange in guinea pig airway smooth muscle and is neuroprotective against glutamate/NMDA toxicity.PPADS tetrasodiuma inhibits P2X1, P2X-2, P2X-3, and P2X- 5. 5.

        Product detail

      • Ppc-1

        Ref: T16565
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        Ppc-1 (Legacy Tebubio ref. 282T16565). Ppc-1 is a chemical compound known for its inhibitory effects on the Gram-negative periodontopathogen Porphyromonas gingivalis. It acts as a mitochondrial uncoupler, enhancing mitochondrial oxygen consumption without affecting ATP production. Additionally, Ppc-1 serves as a cell-permeate inhibitor of interleukin-2 (IL-2). This compound exhibits various beneficial activities, including anti-obesity, antibacterial, and anti-inflammatory properties.

        Product detail

      • Propyl pyrazole triol

        Ref: T16566
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €44.00

        Propyl pyrazole triol (Legacy Tebubio ref. 282T16566). Propyl pyrazole triol (PPT) is a selective agonist of estrogen receptor alpha (ERα), exhibiting a relative binding affinity of 49% for ERα, which is approximately 410 times higher than its affinity for estrogen receptor beta (ERβ: 0.12%).

        Product detail

      • PQR530

        Ref: T16567
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €33.00

        PQR530 (Legacy Tebubio ref. 282T16567). PQR530 is a highly potent dual pan-PI3K/mTORC1/2 inhibitor. PQR530 inhibited protein kinase B (PKB, pSer473) and ribosomal protein S6 (pS6, pSer235/236) phosphorylation with IC50 values of 0.07 μM. It also showing antitumor activity.

        Product detail

      • PR-924

        Ref: T16568
        Sizes: 2 mg, 1 mL * 10 mM (in DMSO)
        From: €820.00

        PR-924 (Legacy Tebubio ref. 282T16568). PR-924 is a selective inhibitor of tripeptide epoxyketone immunoproteasome subunit LMP-7 (IC50: 22 nM). PR-924 inhibits growth and triggers apoptosis in multiple myeloma (MM) cells. PR-924 has antitumor activities. PR-924 covalently modifies proteasomal N-terminal threonine active sites.

        Product detail