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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70846 )

      • Fludrocortisone

        Ref: T1666L
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €40.00

        Fludrocortisone (Legacy Tebubio ref. 282T1666L). Fludrocortisone （Florinef） is a synthetic corticosteroid with moderate glucocorticoid potency and greater mineralocorticoid potency. Fludrocortisone is in research use for the treatment of hypotension.[3]

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      • Tandutinib

        Ref: T1667
        Sizes: 25 mg, 100 mg, 50 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €44.00

        Tandutinib (Legacy Tebubio ref. 282T1667). Tandutinib (CT53518) (MLN518, CT53518), an effective FLT3 antagonist (IC50: 0.22 μM), can also inhibit c-Kit and PDGFR, 15-20 fold higher potency for FLT3 versus CSF-1R and >100-fold selectivity for the same target versus FGFR, EGFR, and KDR.

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      • PS210

        Ref: T16670
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €36.00

        PS210 (Legacy Tebubio ref. 282T16670). PS210 is a potent and selective activator of PDK1 (Kd: 3 μM), specifically targeting the PIF-binding pocket of PDK1 without affecting other protein kinases such as S6K, PKB/Akt, or GSK3. Its prodrug, PS423, serves as a substrate-selective inhibitor of PDK1 in cells, inhibiting the phosphorylation and activation of S6K.

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      • PS315

        Ref: T16671
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        PS315 (Legacy Tebubio ref. 282T16671). PS315 inhibits the full-length and catalytic domain constructs of PKCζ (IC50=10 μM) and PKCη (IC50=30 μM). PS315 has anti-cancer activity. PS315 is a derivative of PS48 and is an allosteric PKC inhibitor by binding to the PIF-pocket of aPKC and inducing displacement of the active site residue Lys111.

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      • PSB-1114 tetrasodium

        Ref: T16672
        Sizes: 500 μg
        From: €926.00

        PSB-1114 tetrasodium (Legacy Tebubio ref. 282T16672). PSB-1114 tetrasodium shows >50-fold selectivity versus the P2Y4 (EC50: 9.3 μM) and P2Y6 (EC50: 7.0 μM) receptors. PSB-1114 tetrasodium is an effective, enzymatically stable, and subtype-selective P2Y2 receptor agonist (EC50: 134 nM) .

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      • Pseudouridimycin

        Ref: T16673
        Sizes: 10 mg
        Price Enquiry

        Pseudouridimycin (Legacy Tebubio ref. 282T16673). Pseudouridimycin is a C-nucleoside analogue. Pseudouridimycin is an antibiotic and is a selective bacterial RNA polymerase (RNAP) inhibitor. It is effective against both Gram-negative and Gram-positive bacteria.

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      • Pseudouridine

        Ref: T16674
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €35.00

        Pseudouridine (Legacy Tebubio ref. 282T16674). Pseudouridine is the most abundant modified nucleoside in non-coding RNAs. It enhances the function of transfer RNA and ribosomal RNA by stabilizing RNA structure.

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      • PSI-697

        Ref: T16676
        Sizes: 25 mg, 100 mg, 50 mg, 1 mL * 10 mM (in DMSO)
        From: €316.00

        PSI-697 (Legacy Tebubio ref. 282T16676). PSI-697 (P-Selectin Inhibitor) is an orally active P-selectin inhibitor with anti-inflammatory and anti-thrombotic effects, useful for studying cardiovascular diseases such as atherosclerosis.

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      • Psicofuranine

        Ref: T16677
        Sizes: 5 mg
        Price Enquiry

        Psicofuranine (Legacy Tebubio ref. 282T16677). Psicofuranine also specifically inhibits GMP synthase and interrupts parasite growth. Psicofuramine is a nucleoside antibiotic. It has the inhibition of xanthosine 5'-phosphate aminase. Psicofuranine shows dose-dependent inhibition of P. falciparum growth(IC50: 0.3 mM).

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