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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70847 )

      • Razuprotafib

        Ref: T16724
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €288.00

        Razuprotafib (Legacy Tebubio ref. 282T16724). Razuprotafib (AKB-9778) is a protein tyrosine phosphatase ß (HPTPß) inhibitor with an IC50 of 50 nM. It effectively activates Tie-2 and provides protection against acute kidney injury.

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      • RCM-1

        Ref: T16725
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €44.00

        RCM-1 (Legacy Tebubio ref. 282T16725). RCM-1 is an inhibitor of FOXM1.

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      • Rebeccamycin

        Ref: T16726
        Sizes: 500 μg, 2500 μg
        From: €506.00

        Rebeccamycin (Legacy Tebubio ref. 282T16726). Rebeccamycin is an antitumor antibiotic+ inhibits DNA topoisomerase I. Rebeccamycin appears to exert its primary antineoplastic effect by poisoning topoisomerase I. It also has a negligible effect on protein kinase C and topoisomerase II.

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      • Relacorilant

        Ref: T16727
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €129.00

        Relacorilant (Legacy Tebubio ref. 282T16727). Relacorilant is a selective and orally bioavailable antagonist of glucocorticoid receptor(Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively). Relacorilant has the potential for Cushing’s syndrome treatment.

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      • Reldesemtiv

        Ref: T16728
        Sizes: 1 mg, 5 mg, 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €167.00

        Reldesemtiv (Legacy Tebubio ref. 282T16728). Reldesemtiv (CK-2127107) is a selective fast skeletal muscle troponin activator with an EC50 of 3.4 μM, enhancing exercise performance in heart failure models.

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      • Remetinostat

        Ref: T16729
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €49.00

        Remetinostat (Legacy Tebubio ref. 282T16729). Remetinostat (SHP-141), a hydroxamic acid-based inhibitor of histone deacetylase enzymes, is currently being developed for the treatment of cutaneous T-cell lymphoma.

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      • Acamprosate calcium

        Ref: T1673
        Sizes: 25 mg, 50 mg, 1 mL * 10 mM (in H2O)
        From: €35.00

        Acamprosate calcium (Legacy Tebubio ref. 282T1673). Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.

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      • Remibrutinib

        Ref: T16730
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €112.00

        Remibrutinib (Legacy Tebubio ref. 282T16730). Remibrutinib inhibits BTK activity with an IC50 value of 0.023 μM in blood. Remibrutinib is an effective and orally active Bruton tyrosine kinase inhibitor (IC50: 1 nM). Remibrutinib has the potential for Chronic urticaria (CU) treatment.

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      • Rentiapril racemate

        Ref: T16731
        Sizes: 1 mg
        From: €137.00

        Rentiapril racemate (Legacy Tebubio ref. 282T16731). Rentiapril racemate (SA-446 racemate) is the racemic form of Rentiapril, exhibiting anti-inflammatory properties and potential applications in glaucoma research.

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