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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70851 )

      • Rigosertib

        Ref: T16750
        Sizes: 5 mg, 10 mg, 2 mg
        From: €39.00

        Rigosertib (Legacy Tebubio ref. 282T16750). Rigosertib (ON-01910) is a selective, non-ATP-competitive PLK1 inhibitor (IC50: 9 nM) and multi-kinase inhibitor. As a selective anti-cancer agent, Rigosertib induces apoptosis by inhibiting the PI3 kinase/Akt pathway, promotes histone H2AX phosphorylation, and induces G2/M arrest in the cell cycle.

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      • Rilapladib

        Ref: T16751
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €107.00

        Rilapladib (Legacy Tebubio ref. 282T16751). Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2, IC50 = 230 pM) and acts as an antagonist of the platelet-activating factor receptor.

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      • Rimacalib

        Ref: T16752
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        Rimacalib (Legacy Tebubio ref. 282T16752). Rimacalib is an inhibitor of Ca2+/calmodulin-dependent protein kinase II (IC50s: ~1 μM for CaMKIIα and ~30 μM for CaMKIIγ).

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      • RIP2 kinase inhibitor 2

        Ref: T16753
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €223.00

        RIP2 kinase inhibitor 2 (Legacy Tebubio ref. 282T16753). RIP2 kinase inhibitor 2 is a compound that inhibits receptor-interacting protein-2 kinase (RIP2).

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      • RIPGBM

        Ref: T16754
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €37.00

        RIPGBM (Legacy Tebubio ref. 282T16754). RIPGBM is a selective inducer of apoptosis in glioblastoma multiforme cancer stem cells (EC50: ≤500 nM).

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      • RIPK-IN-4

        Ref: T16755
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,624.00

        RIPK-IN-4 (Legacy Tebubio ref. 282T16755). RIPK-IN-4 is an effective and selective inhibitor of RIPK2. It also has excellent oral bioavailability (IC50: 3 nM).

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      • Risarestat

        Ref: T16756
        Sizes: 1 mg, 5 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €188.00

        Risarestat (Legacy Tebubio ref. 282T16756). Risarestat (CT-112) is a potent aldose reductase inhibitor and thyroid hormone receptor (TR) antagonist for the treatment of hypoglycemia.

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      • Risdiplam

        Ref: T16757
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg
        From: €63.00

        Risdiplam (Legacy Tebubio ref. 282T16757). Risdiplam (RG7916) is a centrally and peripherally distributed and orally administrable small molecule SMN2 pre-mRNA splicing modifier that increases survival motor neuron (SMN) protein levels.

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      • Rispenzepine

        Ref: T16758
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        Rispenzepine (Legacy Tebubio ref. 282T16758). Rispenzepine is a novel antagonist of muscarinic acetylcholine receptors (mAChRs), selectively targeting the M1 and M3 receptor subtypes, and can be used in the treatment of immune system disorders, infections, and respiratory diseases.

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