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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70851 )

      • Ritanserin

        Ref: T16759
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €39.00

        Ritanserin (Legacy Tebubio ref. 282T16759). Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist with an IC50 of 0.9 nM.

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      • Rosuvastatin

        Ref: T1676
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: €52.00

        Rosuvastatin (Legacy Tebubio ref. 282T1676). Rosuvastatin (ZD4522) is an inhibitor of HMG-CoA reductase (HMGCR) (IC50=11 nM), selective and competitive. Rosuvastatin has hypolipidemic and antiatherosclerotic effects.

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      • RK-24466

        Ref: T16760
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €69.00

        RK-24466 (Legacy Tebubio ref. 282T16760). RK-24466 (KIN 001-51) is a selective and potent Lck inhibitor, targeting Lck (64-509) and LckCD isoforms with IC50 values of less than 1 nM and 2 nM, respectively.

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      • RK-287107

        Ref: T16761
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €39.00

        RK-287107 (Legacy Tebubio ref. 282T16761). RK-287107 is an effective and specific inhibitor of tankyrase (IC50s: 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively).

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      • RMC-4550

        Ref: T16762
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €64.00

        RMC-4550 (Legacy Tebubio ref. 282T16762). RMC-4550 is an effective and allosteric inhibitor of SHP2 (IC50: 0.583 nM).

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      • RN-1747

        Ref: T16763
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €42.00

        RN-1747 (Legacy Tebubio ref. 282T16763). RN-1747 is a selective transient receptor potential cation channel subfamily V member 4 agonist (EC50: hTRPV4 of 0.77 μM, mTRPV4 of 4.0 μM, and rTRPV4 of 4.1 μM) and also acts as an antagonist for TRPM8 (IC50: 4 μM).

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      • RN-18

        Ref: T16764
        Sizes: 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €33.00

        RN-18 (Legacy Tebubio ref. 282T16764). RN-18 is an inhibitor of HIV-1 viral infectivity factor (IC50: 6 μM in nonpermissive H9 cells).

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      • RNPA1000

        Ref: T16765
        Sizes: 100 mg, 50 mg
        From: €831.00

        RNPA1000 (Legacy Tebubio ref. 282T16765). RNPA1000 is an attractive antimicrobial development candidate and RnpA inhibitor.

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      • Ro 08-2750

        Ref: T16766
        Sizes: 5 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €71.00

        Ro 08-2750 (Legacy Tebubio ref. 282T16766). Ro 08-2750 is a non-peptide, reversible nerve growth factor (NGF) inhibitor that binds to NGF with an IC50 of approximately 1 µM. It is also a selective MSI RNA-binding activity inhibitor, exhibiting an IC50 of 2.7 μM. Additionally, Ro 08-2750 selectively inhibits NGF binding to p75NTR over TRKA.

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