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    Results for Activators & Inhibitors ( 70851 )

      • Ref: T16798
        Sizes: 5 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €39.00

        RS 17053 hydrochloride (Legacy Tebubio ref. 282T16798). RS 17053 hydrochloride is a potent and selective antagonist of the α1A adrenoceptor, with a pKi value of 9.1 in native cell membranes and a pA2 value of 9.8 in functional assays.

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      • Ref: T16799
        Sizes: 25 mg, 100 mg, 50 mg, 1 mL * 10 mM (in DMSO)
        From: €415.00

        RS-246204 (Legacy Tebubio ref. 282T16799). RS-246204 is an R-spondin-1 substitute compound. RS-246204 is able to initiate small intestinal organoids without the use of the R-spondin-1 protein.

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      • Ref: T1680
        Sizes: 1 g, 10 g, 5 g, 1 mL * 10 mM (in DMSO)
        From: €46.00

        Tolazoline hydrochloride (Legacy Tebubio ref. 282T1680). Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn.

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      • Ref: T16800
        Sizes: 25 mg, 100 mg, 50 mg
        From: €4,279.00

        (RS)-AMPA (Legacy Tebubio ref. 282T16800). (RS)-AMPA ((±)-AMPA) is a glutamate analog and an agonist of the effective and selective excitatory neurotransmitter L-glutamic acid.

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      • Ref: T16801
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: €41.00

        (RS)-(Tetrazol-5-yl)glycine (Legacy Tebubio ref. 282T16801). (RS)-(Tetrazol-5-yl)glycine (LY 285265) [(D,L-(tetrazol-5-yl)glycine] is an effective and selective N-methyl-D-aspartate receptor agonist with EC50s of 99 nM for GluN1/GluN2D and 1.7 μM for GluN1/GluN2A.

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      • Ref: T16802
        Sizes: 1 mg, 5 mg, 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €204.00

        Lonapalene (Legacy Tebubio ref. 282T16802). Lonapalene (RS4317) is a 5-lipoxygenase (5-LO) inhibitor with anti-psoriasis efficacy.Lonapalene topically blocks skin inflammation.

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      • Ref: T16803
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €84.00

        RS 8359 (Legacy Tebubio ref. 282T16803). RS 8359 is a reversible inhibitor of monoamine oxidase A (MAO-A) with a selectivity ratio of about 2200 for the A:B enzyme types. RS 8359 has antidepressant activity.

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      • Ref: T16805
        Sizes: 25 mg, 100 mg, 50 mg
        From: €2,236.00

        RTS-V5 (Legacy Tebubio ref. 282T16805). RTS-V5 is a dual inhibitor of HDAC/proteasome (IC50s: 6.9, 18, 15, 0.27, 0.53 μM for HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, respectively).

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      • Ref: T16806
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €41.00

        RU-302 (Legacy Tebubio ref. 282T16806). RU-302 is a pan inhibitor of TAM Receptor blocking the interface between the TAM Ig1 ectodomain and the Gas6 Lg domain. RU-302 effectively blocks the activation of Gas6-inducible AXL and suppresses lung cancer tumor growth.

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