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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70864 )

      • Methacholine Chloride

        Ref: T1682
        Sizes: 100 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €54.00

        Methacholine Chloride (Legacy Tebubio ref. 282T1682). Methacholine Chloride (Acetyl-β-methylcholine chloride) is a quaternary ammonium parasympathomimetic agent with the muscarinic actions of ACETYLCHOLINE. It is hydrolyzed by ACETYLCHOLINESTERASE at a considerably slower rate than ACETYLCHOLINE and is more resistant to hydrolysis by nonspecific CHOLINESTERASES so that its actions are more prolonged. It is used as a parasympathomimetic bronchoconstrictor agent and as a diagnostic aid for bronchial asthma.

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      • Actriol

        Ref: T1683
        Sizes: 1 mg, 5 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €55.00

        Actriol (Legacy Tebubio ref. 282T1683). Actriol (Epiestriol) is always used as Glucocorticoid Receptor agonist.

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      • S-MTC

        Ref: T16830
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        S-MTC (Legacy Tebubio ref. 282T16830). S-MTC is a selective inhibitor of type I nitric oxide synthase.

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      • (S)-SNAP5114

        Ref: T16831
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €35.00

        (S)-SNAP5114 (Legacy Tebubio ref. 282T16831). (S)-SNAP5114 is a selective inhibitor of GABA transport, exhibiting IC50 values of 5 μM for hGAT-3 and 21 μM for rGAT-2, and possesses anticonvulsant properties.

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      • S18-000003

        Ref: T16832
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €60.00

        S18-000003 (Legacy Tebubio ref. 282T16832). S18-000003 is an effective orally bioavailable retinoic acid receptor-related orphan receptor-gamma-t inhibitor (IC50: 29 nM). S18-000003 inhibits IL-17 production.

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      • S1P1 Agonist III

        Ref: T16833
        Sizes: 100 mg
        From: €1,019.00

        S1P1 Agonist III (Legacy Tebubio ref. 282T16833). S1P1 Agonist III is an effective and orally active S1P1 agonist (EC50: 18 nM).

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      • S26131

        Ref: T16834
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €41.00

        S26131 (Legacy Tebubio ref. 282T16834). S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of 0.5 and 112 nM respectively.

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      • SAFit1

        Ref: T16835
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,589.00

        SAFit1 (Legacy Tebubio ref. 282T16835). SAFit1 is an inhibitor of FK506 binding protein 51 (FKBP51)-specific (Ki: 4±0.3 nM).

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      • SAFit2

        Ref: T16836
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €112.00

        SAFit2 (Legacy Tebubio ref. 282T16836). SAFit2 is a highly potent and selective inhibitor of fk506 binding protein 51 (FKBP51) with a Ki value of 6 nM. SAFit2 can enhance the binding of AKT2-AS160 and participate in the downstream response of glucocorticoid release in vivo. It is a candidate compound for the treatment of obesity, chronic pain, depression and anxiety.

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