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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70864 )

      • Sarolaner

        Ref: T16845
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €50.00

        Sarolaner (Legacy Tebubio ref. 282T16845). Sarolaner (PF-6450567) is an orally active, broad-spectrum ectoparasiticide with an LC80 of 0.3 μg/mL against C. felis and an LC100 of 0.003 μg/mL against O. turicata.

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      • Sauristolactam

        Ref: T16846
        Sizes: 25 mg
        Price Enquiry

        Sauristolactam (Legacy Tebubio ref. 282T16846). Sauristolactam inhibits the receptor activator of nuclear factor-κB ligand (RANKL)-induced osteoclastogenesis and has the potential to inhibit osteoclast differentiation. Sauristolactam, a natural aristolactam isolated from aerial portions of Saururus Chinensis. Sauristolactam has significant neuroprotective activity against glutamate-induced toxicity in primary cultured rat cortical cells.

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      • SB-218078

        Ref: T16848
        Sizes: 1 mg
        From: €401.00

        SB-218078 (Legacy Tebubio ref. 282T16848). SB-218078 is less potently inhibits Cdc2 (IC50: 250 nM) and PKC (IC50: 1000 nM). SB-218078 is a potent, ATP-competitive, and cell-permeable checkpoint kinase 1 inhibitor that inhibits Chk1 phosphorylation of cdc25C (IC50: 15 nM).

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      • SB-222200

        Ref: T16849
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €38.00

        SB-222200 (Legacy Tebubio ref. 282T16849). SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).

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      • 2-Amino-5-chlorobenzophenone

        Ref: T1685
        Sizes: 1 g, 100 mg, 50 mg, 500 mg, 1 mL * 10 mM (in DMSO)
        From: €39.00

        2-Amino-5-chlorobenzophenone (Legacy Tebubio ref. 282T1685). 2-Amino-5-chlorobenzophenone is used as pharmaceutical intermediates.

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      • SB-265610

        Ref: T16850
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €58.00

        SB-265610 (Legacy Tebubio ref. 282T16850). SB-265610 (GSK-CXCR2) is a nonpeptide and allosteric CXCR2 antagonist. SB-265610 blocks rat cytokine-induced neutrophil chemoattractant-1 (CINC-1)-induced calcium mobilization and neutrophil chemotaxis (IC50s: 3.7 nM and 70 nM, respectively).

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      • SB-267268

        Ref: T16851
        Sizes: 25 mg, 100 mg, 50 mg
        From: €2,236.00

        SB-267268 (Legacy Tebubio ref. 282T16851). SB-267268 inhibits human and mouse αvβ3 (IC50s: 0.68 and 0.29 nM, respectively). SB-267268 is a selective and nonpeptidic alpha(v)beta3 and alpha(v)beta5 integrins antagonist (Kis: 0.9, 0.5 and 0.7 nM for human αvβ3, monkey αvβ3 and human αvβ5, respectively).

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      • SB-568849

        Ref: T16852
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,896.00

        SB-568849 (Legacy Tebubio ref. 282T16852). SB-568849 is an antagonist of the melanin-concentrating hormone receptor 1 (pKi: 7.7).

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      • SB-633825

        Ref: T16853
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 2 mg
        From: €223.00

        SB-633825 (Legacy Tebubio ref. 282T16853). SB-633825 can inhibit cancer cell growth and angiogenesis. SB-633825 is an effective and ATP-competitive inhibitor of TIE2, LOK, and BRK (IC50s: 3.5 nM, 66 nM, 150 nM, respectively).

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