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    Results for Activators & Inhibitors ( 107980 )

      • Ref: T10142
        Sizes: 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €39.00

        p-Ethynylphenylalanine (Legacy Tebubio ref. 282T10142). p-Ethynylphenylalanine (4-Ethynyl-L-phenylalanine), a selective, effective, and reversible tryptophan hydroxylase (TPH) inhibitor, exhibits competitive inhibition with a Ki of 32.6 μM.

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      • Ref: T10142L
        Sizes: 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €35.00

        p-Ethynylphenylalanine hydrochloride (Legacy Tebubio ref. 282T10142L). p-Ethynylphenylalanine hydrochloride (4-Ethynyl-L-phenylalanine HCL) is a novel, potent, and specific inhibitor of TPH[1]. Its potential to selectively and reversibly inhibit serotonin biosynthesis may contribute to characterizing the role of serotonin in behavioral and physiological activities[1].

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      • Ref: T10144
        Sizes: 1 mg, 5 mg
        From: €415.00

        4-Hydroxyatomoxetine D3 (Legacy Tebubio ref. 282T10144). 4-Hydroxyatomoxetine D3 is a deuterium labeled 4-Hydroxyatomoxetine. 4-Hydroxyatomoxetine is an active metabolite of Atomoxetine. 4-Hydroxyatomoxetine is metabolized by CYP2D6. Atomoxetine is a noradrenaline reuptake inhibitor.

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      • Ref: T10146
        Sizes: 1 mg, 5 mg, 25 mg, 10 mg
        From: €139.00

        4-Hydroxyderricin (Legacy Tebubio ref. 282T10146). 4-Hydroxyderricin, a potent and selective MAO-B inhibitor (IC50: 3.43 μM), is the main active ingredient of Angelica sinensis, which mildly inhibits dopamine β-hydroxylase (DBH) activity and possesses antidepressant activity.

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      • Ref: T10147
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €45.00

        4-Hydroxymephenytoin (Legacy Tebubio ref. 282T10147). 4-Hydroxymephenytoin ((+/-)-4'-Hydroxymephenytoin) is the metabolism of an antiepileptic drug mephenytoin. Mephenytoin is used as a CYP2C19 substrate.

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      • Ref: T10148
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €55.00

        4-Hydroxynonenal (Legacy Tebubio ref. 282T10148). 4-Hydroxynonenal (4-HNE) (4-HNE) is an oxidative/nitrosative stress biomarker. It is a substrate and an inhibitor of acetaldehyde dehydrogenase 2 (ALDH2).

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      • Ref: T10149
        Sizes: 1 mg, 5 mg
        From: €259.00

        4-Hydroxypropranolol-d7 hydrochloride (Legacy Tebubio ref. 282T10149). 4-Hydroxypropranolol D7 hydrochloride is deuterium-labeled 4-Hydroxypropranolol hydrochloride. 4-Hydroxypropranolol hydrochloride is an active metabolite of Propranolol, with a potency comparable to Propranolol. It inhibits β1- and β2-adrenergic receptors (pA2s: 8.24 and 8.26).

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      • Ref: T10151
        Sizes: 25 mg, 100 mg, 50 mg
        From: €2,123.00

        5-Lipoxygenase-In-1 (Legacy Tebubio ref. 282T10151). 5-Lipoxygenase-In-1 (compound example 4.10) is a 5-Lipoxygenase inhibitor.

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      • Ref: T10152
        Sizes: 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €37.00

        4-Methylamino antipyrine (Legacy Tebubio ref. 282T10152). 4-Methylamino antipyrine, an active metabolite of Metamizole, a pyrazolone non-steroidal anti-inflammatory drug (NSAID) that inhibits COX, possesses analgesic, antipyretic, and relatively weak anti-inflammatory properties.

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