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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 107979 )

      • Fluorothyl

        Ref: T1017
        Sizes: 100 mg, 50 mg, 500 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €38.00

        Fluorothyl (Legacy Tebubio ref. 282T1017). Fluorothyl (Bis(2,2,2-trifluoroethyl) ether) is a convulsant used in experimental animals.

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      • 5-HT7 agonist 1

        Ref: T10170
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €133.00

        5-HT7 agonist 1 (Legacy Tebubio ref. 282T10170). 5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM). 5-HT7 agonist 1 can be used in studies about CNS disorders.

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      • 5-Hydroxypyrazine-2-Carboxylic Acid

        Ref: T10171
        Sizes: 500 mg
        From: €48.00

        5-Hydroxypyrazine-2-Carboxylic Acid (Legacy Tebubio ref. 282T10171). 5-Hydroxypyrazine-2-Carboxylic Acid is a metabolite of anti-tuberculosis drug pyrazinamide.

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      • 5-Iodo-indirubin-3'-monoxime

        Ref: T10172
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg
        From: €338.00

        5-Iodo-indirubin-3'-monoxime (Legacy Tebubio ref. 282T10172). 5-Iodo-indirubin-3'-monoxime is a potent inhibitor of GSK-3β, CDK5/P25, and CDK1/cyclin B, competing with ATP for binding to the catalytic site of the kinase (IC50s: 9, 20, and 25 nM).

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      • MCHR1 antagonist 1

        Ref: T10173
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        MCHR1 antagonist 1 (Legacy Tebubio ref. 282T10173). MCHR1 antagonist 1 is a selective antagonist of the melanin-concentrating hormone-1 (MCH1) receptor with a Kb of 1 nM and a Ki of 4 nM at the human MCH1 receptor.

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      • 5-R-Rivaroxaban

        Ref: T10174
        Sizes: 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €35.00

        5-R-Rivaroxaban (Legacy Tebubio ref. 282T10174). 5-R-Rivaroxaban is the (R)-enantiomer of Rivaroxaban. Rivaroxaban (BAY 59-7939) is a highly potent and selective direct Factor Xa (FXa) inhibitor with an IC50 of 0.7 nM and a Ki of 0.4 nM.

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      • TRPV antagonist 1

        Ref: T10176
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        TRPV antagonist 1 (Legacy Tebubio ref. 282T10176). TRPV antagonist 1 is an antagonist of transient receptor potential vanilloid (TRPV; IC50 < 250 nM).

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      • (5Z,2E)-CU-3

        Ref: T10177
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €47.00

        (5Z,2E)-CU-3 (Legacy Tebubio ref. 282T10177). (5Z,2E)-CU-3 is a potent and highly selective inhibitor of the DGKα isozyme with an IC50 value of 0.6 μM, competing with ATP and exhibiting a Km value of 0.48 mM. It specifically targets the catalytic region of DGKα without affecting the regulatory region and has demonstrated antitumor and immunogenic effects by promoting cancer cell apoptosis and T cell activation.

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      • 5β-​Dutasteride

        Ref: T10179
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        5β-​Dutasteride (Legacy Tebubio ref. 282T10179). 5β-Dutasteride (5β, S-configuration of Dutasteride) is a potent inhibitor of both 5 alpha-reductase isozymes.

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