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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 107979 )

      • PDE IV-IN-1

        Ref: T10201
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €408.00

        PDE IV-IN-1 (Legacy Tebubio ref. 282T10201). PDE IV-IN-1 is a potent phosphodiesterase 4 (PDE4) inhibitor with anti-inflammatory activity for the treatment of asthma, chronic obstructive pulmonary disease and other inflammatory diseases, and is a potential compound for the study of depression.

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      • A 1070722

        Ref: T10202
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €44.00

        A 1070722 (Legacy Tebubio ref. 282T10202). A 1070722 is a potent and selective GSK-3 inhibitor, exhibiting high affinity for both GSK-3α (Ki = 0.6 nM) and GSK-3β (Ki = 0.6 nM). It can penetrate the blood-brain barrier (BBB) and accumulate in brain regions, indicating potential use as a PET radiotracer for quantifying GSK-3 in the brain.

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      • A 1120

        Ref: T10203
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €44.00

        A 1120 (Legacy Tebubio ref. 282T10203). A 1120 is a nonretinoid retinol-binding protein 4 (RBP4) antagonist (Ki: 8.3 nM), which disrupts the interaction between RBP4 and its binding partner transthyretin.

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      • A-317491 sodium salt hydrate

        Ref: T10204
        Sizes: 5 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        Price Enquiry

        A-317491 sodium salt hydrate (Legacy Tebubio ref. 282T10204). A-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist that inhibits receptor-mediated calcium flux.

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      • A-395

        Ref: T10205
        Sizes: 1 mg, 5 mg, 25 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €46.00

        A-395 (Legacy Tebubio ref. 282T10205). A-395 is an antagonist of polycomb repressive complex 2 (PRC2) protein-protein interactions that potently inhibits the trimeric PRC2 complex (EZH2-EED-SUZ12, IC50: 18 nM).

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      • A 419259

        Ref: T10206
        Sizes: 2 mg
        From: €77.00

        A 419259 (Legacy Tebubio ref. 282T10206). A 419259 is a pyrrolo-pyrimidine inhibitor, designed to enhance selectivity towards the Src family (IC50s: 9 nM, <3 nM and <3 nM for Src, Lck and Lyn).

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      • A 438079

        Ref: T10207
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €47.00

        A 438079 (Legacy Tebubio ref. 282T10207). A 438079 is a potent and selective antagonist of the P2X7 receptor (pIC50: 6.9).

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      • A-69412

        Ref: T10208
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €133.00

        A-69412 (Legacy Tebubio ref. 282T10208). A-69412 (N-1-(Fur-3-ylethyl)-N-hydroxyurea) is a reversible, specific inhibitor of the hydrophilic 5-lipoxygenase. It has the potential to treat ulcerative colitis and asthma, and possibly other inflammatory and allergic conditions.

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      • (R)-Lansoprazole

        Ref: T1021
        Sizes: 100 mg, 50 mg, 500 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €38.00

        (R)-Lansoprazole (Legacy Tebubio ref. 282T1021). (R)-Lansoprazole (T 168390) is the R-isomer of lansoprazole and a substituted benzimidazole prodrug with selective and irreversible proton pump inhibitor activity.Lansoprazole (AG 1749) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor (exosome inhibitor)

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