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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 107979 )

      • A-9758

        Ref: T10210
        Sizes: 25 mg, 100 mg, 50 mg
        From: €2,917.00

        A-9758 (Legacy Tebubio ref. 282T10210). A-9758 is a RORγ ligand and selective RORγt inverse agonist (IC50: 5 nM) that effectively suppresses IL-17A release, Th17 differentiation, and Th17 effector function, significantly attenuating IL-23 driven psoriasiform dermatitis.

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      • Aβ42-IN-1

        Ref: T10211
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        Aβ42-IN-1 (Legacy Tebubio ref. 282T10211). Aβ42-IN-1, compound 1v, is a novel, potent and orally active γ-secretase modulator (GSM). Aβ42-IN-1 potently reduced Aβ42 levels with an IC 50 value of 0.091 μM in cultured cells without inhibiting CYP3A4. Aβ42-IN-1 shows a sustained pharmacokinetic profile.

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      • A2AR-agonist-1

        Ref: T10212
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €111.00

        A2AR-agonist-1 (Legacy Tebubio ref. 282T10212). A2AR-agonist-1 (N-(2-(1H-Indol-3-yl)ethyl)adenosine) is a potent A2AR and ENT1 agonist (Ki: 4.39 and 3.47 for A2AR and ENT1. It targets the Adenosine A2A Receptor and Adenosine Transporter for Neuroprotection.

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      • A-437203

        Ref: T10213
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €104.00

        A-437203 (Legacy Tebubio ref. 282T10213). A-437203 (Lu201640) is A kind of based on 1 h - pyrimidin - 2 - one sca ff old, selective, new powerful d3 receptor antagonist, on D2, d3, and D4 receptor, Ki value 71, respectively 1.6 and 6220 nM.

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      • A7132

        Ref: T10214
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 500 mg, 10 mg
        From: €398.00

        A7132 (Legacy Tebubio ref. 282T10214). A7132 is an antibacterial agent and possesses broad and potent antibacterial activity.

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      • AAPK-25

        Ref: T10215
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €99.00

        AAPK-25 (Legacy Tebubio ref. 282T10215). AAPK-25 is a potent and selective Aurora/PLK dual inhibitor with anti-tumor activity, causing mitotic delay and arresting cells in prometaphase, followed by increased apoptosis. It targets Aurora-A/-B/-C with Kd values ranging from 23-289 nM.

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      • AB-680

        Ref: T10216
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €131.00

        AB-680 (Legacy Tebubio ref. 282T10216). AB-680, a highly potent, reversible, and selective inhibitor of CD73 (an ectonucleotidase, Ki: 4.9 pM for hCD73) with anti-tumor activity, displays >10,000-fold selectivity over related ectonucleotidases CD39.

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      • Abarelix Acetate (183552-38-7 free base)

        Ref: T10217
        Sizes: 5 mg, 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        Price Enquiry

        Abarelix Acetate (183552-38-7 free base) (Legacy Tebubio ref. 282T10217). Abarelix (PPI 149; R 3827) Acetate is a potent gonadotrophin-releasing hormone (GnRH) antagonist, used for prostate cancer research.

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      • Abarelix

        Ref: T10217L
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €40.00

        Abarelix (Legacy Tebubio ref. 282T10217L). Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.

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