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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70851 )

      • Methimepip dihydrobromide

        Ref: T37727
        Sizes: 200 mg
        Price Enquiry

        Methimepip dihydrobromide (Legacy Tebubio ref. 282T37727). Methimepip dihydrobromide is a selective H3R agonist.

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      • Methoctramine (hydrate)

        Ref: T37728
        Sizes: 5 mg, 25 mg, 10 mg
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        Methoctramine (hydrate) (Legacy Tebubio ref. 282T37728). Methoctramine is a selective antagonist of M2 muscarinic acetylcholine receptors (IC50 = 6.1 nM in CHO-K1 cell membranes).[1] It is selective for M2 over M1, M3, M4, and M5 receptors (IC50s = 92, 770, 260, and 217 nM, respectively).

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      • IMP-1700

        Ref: T37729
        Sizes: 5 mg, 25 mg, 10 mg
        From: €265.00

        IMP-1700 (Legacy Tebubio ref. 282T37729). IMP-1700 is an inhibitor of bacterial DNA repair.1It potentiates the activity of the quinolone antibiotic ciprofloxacin against methicillin-resistantS. aureus(MRSA) with a combination index value of 0.7. IMP-1700 inhibits the ciprofloxacin-induced bacterial SOS response, a process that repairs DNA damage, in a reporter assay in a concentration-dependent manner. It is also active againstE. coli, as well as methicillin-resistant and -sensitive S. aureus, when used alone (EC50s = 0.5, 0.21, and 3.8 μM, respectively).

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      • Oxypaeoniflorin

        Ref: T3773
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €57.00

        Oxypaeoniflorin (Legacy Tebubio ref. 282T3773). Oxypaeoniflorin a monoterpene glycoside compound isolated from Paeoniae, is an antioxidant, is neuroprotective and anti-inflammatory.

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      • Saccharocarcin A

        Ref: T37730
        Sizes: 2500 μg
        From: €3,315.00

        Saccharocarcin A (Legacy Tebubio ref. 282T37730). Saccharocarcin A is an antibiotic originally isolated from [S. aerocolonigenes subsp. antibiotica]. It demonstrates activity against [M. luteus], [S. aureus], [E. coli], [P. aeruginosa], and [C. albicans] in a disc assay and inhibits [C. trachomatis] infection by 88% without inducing cytotoxicity in McCoy cells at a concentration of 0.5 μg/ml.

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      • TPU-0037A

        Ref: T37731
        Sizes: 5 mg
        Price Enquiry

        TPU-0037A (Legacy Tebubio ref. 282T37731). TPU-0037A is an antibiotic and a congener of lydicamycin. It inhibits the growth of Gram-positive bacteria, including methicillin-resistant S. aureus (MRSA), B. subtilis, and M. luteus (MICs = 1.56-12.5 μg/ml), but not Gram-negative E. coli, P. mirabilis, P. vulgaris, or P. aeruginosa strains (MICs = >50 μg/ml).

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      • AMG 21629

        Ref: T37732
        Sizes: 1 mg
        From: €1,397.00

        AMG 21629 (Legacy Tebubio ref. 282T37732). Potent and selective TRPV1 antagonist. Blocks Ca2+ uptake by CHO cells expressing TRPV1 receptors and acid-induced Ca2+ uptake, respectively). Exhibits >4000-fold selectivity for TRPV1 over other TRP channels. Blocks capsaicin-induced flinch response and causes hyperthermia in rats. Orally available and non-CNS penetrant.

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      • AMP-PNP tetralithium

        Ref: T37733
        Sizes: 10 mg
        From: €964.00

        AMP-PNP tetralithium (Legacy Tebubio ref. 282T37733). Non-hydrolyzable AMP analog. Kir6 (KATP) channel blocker. Inhibits fast axonal transport and stabilizes the interaction of membranous organelles with microtubules.

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      • AMPA receptor modulator-2

        Ref: T37734
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €142.00

        AMPA receptor modulator-2 (Legacy Tebubio ref. 282T37734). AMPA receptor modulator-2 (Example 134) is an AMPA receptor modulator with a pIC50 of 10.1 for TARPγ2 dependent AMPA receptor[1]. pIC50 = -lgIC50. [1]. BERRY CYNTHIA G B (US), et al. AZABENZIMIDAZOLES AND THEIR USE AS AMPA RECEPTOR MODULATORS. Patent. WO2016176460.

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