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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 18112 )

      • BMS202 hydrochloride (1675203-84-5(free base))

        Ref: T4696
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €54.00

        BMS202 hydrochloride (1675203-84-5(free base)) (Legacy Tebubio ref. 282T4696). BMS202 hydrochloride (1675203-84-5(free base)) (PD-1/PD-L1 inhibitor 2 hydrochloride) is a small-molecule PD-1/PD-L1 interaction inhibitor (IC50: 18 nM). Biophysical studies demonstrate that BMS202 binds directly to PD-L1. Binding of BMS202 promotes PD-L1 dimerisation and blocks the PD-L1/ PD1 interaction.

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      • ABBV-744

        Ref: T4697
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €45.00

        ABBV-744 (Legacy Tebubio ref. 282T4697). ABBV-744 is a BDII-selective BET bromodomain inhibitor that inhibits BRD2/3/4. It is used in the research on inflammatory diseases, cancer, and AIDS.

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      • 8-Fluoro-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one

        Ref: T4698
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg
        From: €37.00

        8-Fluoro-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one (Legacy Tebubio ref. 282T4698). 8-Fluoro-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one serves as a pharmaceutical intermediate.

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      • 1,3,5-Trihydroxy-4-prenylxanthone

        Ref: T4700
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        1,3,5-Trihydroxy-4-prenylxanthone (Legacy Tebubio ref. 282T4700). 1,3,5-Trihydroxy-4-prenylxanthone is a relatively potent inhibitor of phosphodiesterase type 5 (PDE5) with an IC50 of 3.0 μM; it exhibits in vitro inhibitory activity against acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) with IC50 values of 56.3plusmn;0.4 and 46.0plusmn;0.3 M, respectively. It also inhibits LPS-induced NF-κB and AP-1 activations by interfering with the posttranslational modification (phosphorylation and/or ubiquitinylation) of IRAK-1, disrupting TAK1-mediated activation of IKK and MAPKs signal transduction.

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      • Diclofop-methyl

        Ref: T4701
        Sizes: 5 mg, 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €46.00

        Diclofop-methyl (Legacy Tebubio ref. 282T4701). Diclofop-methyl is a common post-growth herbicide commonly used in agriculture. It enhances proton permeability of isolated oat root vesicle membranes.

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      • (3-Carboxypropyl)trimethylammonium chloride

        Ref: T4702
        Sizes: 100 mg
        From: €55.00

        (3-Carboxypropyl)trimethylammonium chloride (Legacy Tebubio ref. 282T4702). (3-Carboxypropyl)trimethylammonium chloride ((3-Carboxypropyl)trimethylammonium chlor) is a synthetic carnitine related compound used as a transporter substrate in the cloning and sequencing of human carnitine transporter 2 (CT2).

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      • (2-Aminoethyl)phosphonic acid

        Ref: T4703
        Sizes: 100 mg
        From: €33.00

        (2-Aminoethyl)phosphonic acid (Legacy Tebubio ref. 282T4703). (2-Aminoethyl)phosphonic acid (2-Aminoethylphosphonic acid) is primarily detected in urine. (2-Aminoethyl)phosphonic acid participates in many enzymatic reactions and is also the parent compound of other transformation products, including but not limited to ceramide 2-(methylamino)ethylphosphonate, N-(2-phosphineethyl)cholamide and CMP-2-aminoethylphosphonate.

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      • L-Anserine nitrate

        Ref: T4704
        Sizes: 25 mg, 100 mg, 50 mg, 500 mg, 10 mg
        From: €45.00

        L-Anserine nitrate (Legacy Tebubio ref. 282T4704). L-Anserine nitrate (L-Anserine nitrate salt) is a dipeptide found in most animal tissues. In model systems it is a potent Antioxidant and scavener of hydroxyl radicals. The compound inhibits nonenzymatic protein glycation induced by aldose and ketose reducing sugars. It is much less potent than L-carnosine as an inhibitor of protein crosslinking.

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      • Aminoadipic acid

        Ref: T4705
        Sizes: 1 g, 500 mg, 1 mL * 10 mM (in H2O)
        From: €48.00

        Aminoadipic acid (Legacy Tebubio ref. 282T4705). Aminoadipic acid (DL-2-Aminoadipic acid) (2-aminoadipate) is a metabolite in the principal biochemical pathway of lysine. It is an intermediate in the metabolism (i.e. breakdown or degradation) of lysine and saccharopine. It antagonizes neuroexcitatory activity modulated by the glutamate receptor N-methyl-D-aspartate (NMDA). Aminoadipic acid has also been shown to inhibit the production of kynurenic acid, a broad spectrum excitatory amino acid receptor antagonist, in brain tissue slices.

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