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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70851 )

      • LY2794193

        Ref: T15807
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg
        From: €594.00

        LY2794193 (Legacy Tebubio ref. 282T15807). LY2794193 is a highly effective and selective agonist of the mGlu3 receptor (hmGlu3 Ki=0.927 nM,EC50=0.47 nM; hmGlu2 Ki=412 nM,EC50=47.5 nM).

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      • Merestinib dihydrochloride

        Ref: T15808
        Sizes: 5 mg, 2 mg
        From: €71.00

        Merestinib dihydrochloride (Legacy Tebubio ref. 282T15808). Merestinib dihydrochloride (LY2801653 dihydrochloride) is an orally available kinase inhibitor with antitumor activity that inhibits MET, AXL, RON, and MKNK1/2, and inhibits the growth of NTRK fusion-carrying tumors.

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      • LY2812223

        Ref: T15809
        Sizes: 25 mg, 100 mg, 50 mg
        From: €2,781.00

        LY2812223 (Legacy Tebubio ref. 282T15809). LY2812223 is a highly effective and functionally selective mGlu2 receptor agonist. It has a mGlu2 binding affinity for mGlu2 and mGlu3 (Ki=144 nM and 156 nM, respectively).

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      • Picolamine

        Ref: T1581
        Sizes: 1 g, 1 mL * 10 mM (in DMSO)
        From: €33.00

        Picolamine (Legacy Tebubio ref. 282T1581). Picolamine acts as a potential inhibitor of DPP-4.

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      • LY2922470

        Ref: T15810
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €133.00

        LY2922470 (Legacy Tebubio ref. 282T15810). LY2922470 is a potent, selective G protein-coupled receptor 40 (GPR40) agonist, with EC50s of 7 nM for human GPR40, 1 nM for mouse GPR40 and 3 nM for rat GPR40, respectively. LY2922470 reduces glucose levels along and increases insulin and GLP-1 significantly.

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      • LY2955303

        Ref: T15811
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: €40.00

        LY2955303 (Legacy Tebubio ref. 282T15811). LY2955303 is an effective and selective antagonist of retinoic acid receptor gamma (RARγ, Ki = 1.09 nM).

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      • LY2979165

        Ref: T15812
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg
        From: €78.00

        LY2979165 (Legacy Tebubio ref. 282T15812). LY2979165 (mGlu2 agonist) is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.

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      • LY309887

        Ref: T15813
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,589.00

        LY309887 (Legacy Tebubio ref. 282T15813). LY309887 is a potent inhibitor of glycinamide ribonucleotide formyltransferase (Ki: 6.5 nM) with antitumor activity.

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      • LY3130481

        Ref: T15814
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 1 mL * 10 mM (in DMSO)
        From: €428.00

        LY3130481 (Legacy Tebubio ref. 282T15814). LY3130481 is an AMPA receptor antagonist. It is dependent upon transmembrane AMPA receptor regulatory protein (TARP) γ-8 and selectively inhibits AMPA/TARP γ-8 (IC50: 65 nM).

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