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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70847 )

      • Filorexant

        Ref: T16096
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €35.00

        Filorexant (Legacy Tebubio ref. 282T16096). Filorexant (MK-6096) is an orally bioavailable, effective, and selective reversible antagonist of OX1 and OX2 receptors, with (Ki <3 nM).

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      • MK-8318

        Ref: T16097
        Sizes: 25 mg, 100 mg, 50 mg
        From: €2,577.00

        MK-8318 (Legacy Tebubio ref. 282T16097). MK-8318 is an effective and selective antagonist of the CRTh2 receptor (Ki: 5.0 nM).

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      • Islatravir

        Ref: T16098
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €83.00

        Islatravir (Legacy Tebubio ref. 282T16098). Islatravir (MK-8591) is an effective anti-HIV-1 agent. It acts as a nucleoside reverse transcriptase inhibitor (EC50s: 0.068 nM, 3.1 nM, and 0.15 nM for HIV-1 (WT), HIV-1 (M184V), HIV-1 (MDR), respectively).

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      • MK8722

        Ref: T16099
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €36.00

        MK8722 (Legacy Tebubio ref. 282T16099). MK8722 is an effective and systemic activator of pan-AMPK.

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      • Metaxalone

        Ref: T1610
        Sizes: 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €44.00

        Metaxalone (Legacy Tebubio ref. 282T1610). Metaxalone (Methaxalonum) (marketed by King Pharmaceuticals under the brand name Skelaxin ) is a muscle relaxant used to relax muscles and relieve pain caused by strains, sprains, and other musculoskeletal conditions.

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      • Balamapimod

        Ref: T16100
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        Balamapimod (Legacy Tebubio ref. 282T16100). Balamapimod is a reversible inhibitor of Ras/Raf/MEK. It also has a potential anti-tumor activity.

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      • ML-792

        Ref: T16102
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €96.00

        ML-792 (Legacy Tebubio ref. 282T16102). ML-792 is a specific small ubiquitin-like modifier activating enzyme (SUMO) inhibitor. ML-792 selectively inhibits SAE/SUMO1 and SAE/SUMO2 with IC50 of 3 and 11 nM.

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      • ML-9 Free Base

        Ref: T16103
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        ML-9 Free Base (Legacy Tebubio ref. 282T16103). ML-9 (free base) suppresses MLCK, PKA, and PKC activity (Ki: 4, 32, and 54 μM, respectively). ML-9 (free base) is a selective and effective inhibitor of Akt kinase, inhibits myosin light-chain kinase (MLCK), and stromal interaction molecule 1 (STIM1) activity. ML-9 (free base) causes autophagy by stimulating autophagosome formation and inhibiting their degradation.

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      • ML-9

        Ref: T16104
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €39.00

        ML-9 (Legacy Tebubio ref. 282T16104). ML-9 suppresses MLCK, PKA, and PKC activity with Ki values of 4, 32, and 54 μM, respectively. ML-9 is a selective and effective inhibitor of Akt kinase, inhibits myosin light-chain kinase (MLCK), and stromal interaction molecule 1 (STIM1) activity. ML-9 causes autophagy by stimulating autophagosome formation and inhibiting their degradation.

        Product detail