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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70846 )

      • MSN-125

        Ref: T16155
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        MSN-125 (Legacy Tebubio ref. 282T16155). MSN-125 effectively inhibits Bax/Bak-mediated apoptosis in HCT-116, BMK Cells, and primary cortical neurons protect primary neurons against glutamate excitotoxicity. MSN-125 is an effective Bax and Bak oligomerization inhibitor. MSN-125 prevents mitochondrial outer membrane permeabilization (MOMP) (IC50: 4 μM).

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      • MT 63-78

        Ref: T16156
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg
        From: €89.00

        MT 63-78 (Legacy Tebubio ref. 282T16156). MT 63-78 is a specific and effective direct AMPK activator (EC50: 25 μM) that blocks prostate cancer growth by inhibiting the lipogenesis and mTORC1 pathways. It has antitumor effects and induces cell mitotic arrest and apoptosis.

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      • MT-802

        Ref: T16157
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €100.00

        MT-802 (Legacy Tebubio ref. 282T16157). MT-802 is an effective BTK degrader based on PROTAC technology (DC50: 1 nM). MT-802 has the potential to treat C481S mutant chronic lymphocytic leukemia (CLL).

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      • PF-02575799

        Ref: T16158
        Sizes: 25 mg, 100 mg, 50 mg
        From: €2,066.00

        PF-02575799 (Legacy Tebubio ref. 282T16158). PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).

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      • Muramyl dipeptide

        Ref: T16159
        Sizes: 5 mg, 25 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €235.00

        Muramyl dipeptide (Legacy Tebubio ref. 282T16159). Muramyl dipeptide (MDP) is a synthetic immunoreactive peptide, consisting of N-acetyl muramic acid attached to a short amino acid chain of L-Ala-D-isoGln. It indirectly decreases osteoclast differentiation by reducing the RANKL/OPG ratio and directly increases osteoblast differentiation by up-regulating Runx2 gene expression through MAPK pathways, thereby inducing bone formation via Runx2.

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      • Irbesartan HCl

        Ref: T1615L
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        Irbesartan HCl (Legacy Tebubio ref. 282T1615L). Irbesartan is an angiotensin II receptor antagonist used mainly for the treatment of hypertension. It selectively and competitively blocks the binding of angiotensin II to the angiotensin I receptor.

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      • Cefotiam hydrochloride

        Ref: T1616
        Sizes: 100 mg, 50 mg, 500 mg, 10 mg, 200 mg
        From: €45.00

        Cefotiam hydrochloride (Legacy Tebubio ref. 282T1616). Cefotiam hydrochloride (SCE-963 hydrochloride) is the hydrochloride salt form of cefotiam, a third-generation, semi-synthetic, beta-lactam cephalosporin antibiotic with antibacterial activity. Cefotiam binds to penicillin-binding proteins (PBPs), transpeptidases that are responsible for crosslinking of peptidoglycan. By preventing crosslinking of peptidoglycan, cell wall integrity is lost and cell wall synthesis is halted.

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      • Musk tibetene

        Ref: T16160
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        Musk tibetene (Legacy Tebubio ref. 282T16160). Musk tibetine reveals no genotoxicity in the micronucleus test with human lymphocytes and human hepatoma cell lines. Musk tibetene is a nitro musk compound with carcinogenic activity.

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      • Mutant IDH1 inhibitor

        Ref: T16161
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €40.00

        Mutant IDH1 inhibitor (Legacy Tebubio ref. 282T16161). Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).

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