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Activators & Inhibitors

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    Results for Activators & Inhibitors ( 70847 )

      • Sulbactam

        Ref: T1631
        Sizes: 100 mg, 50 mg, 500 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €44.00

        Sulbactam (Legacy Tebubio ref. 282T1631). Sulbactam (CP45899) is a semi-synthetic beta-lactamase inhibitor. The beta-lactam ring of sulbactam irreversibly binds to beta-lactamase at or near its active site, thereby blocking enzyme activity and preventing metabolism of other beta-lactam antibiotics by the enzyme. Combining this agent with a beta-lactamase susceptible antibiotic, such as penicillins or a cephalosporin, to treat infections caused by beta-lactamase producing organisms, results in a decreased turnover rate of the beta-lactamase sensitive antibiotic and enhances its antibacterial activity.

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      • Sulbactam pivoxil

        Ref: T1631L
        Sizes: 5 mg
        From: €1,101.00

        Sulbactam pivoxil (Legacy Tebubio ref. 282T1631L). Sulbactam pivoxil is an irreversible inhibitor of β-lactamase.

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      • Amitraz

        Ref: T1632
        Sizes: 1 g, 500 mg
        From: €38.00

        Amitraz (Legacy Tebubio ref. 282T1632). Amitraz (NSC 324552) is a white monoclinic crystals. Melting point 187-189°F (86-87°C). Insoluble in water. Used as an acaricide, insecticide and treatment of demodectic mange in dogs.

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      • NI-42

        Ref: T16321
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €44.00

        NI-42 (Legacy Tebubio ref. 282T16321). NI-42 is a structurally orthogonal chemical probe for the BRPFs and is biased. It effective inhibitor of the BRD of the BRPFs (IC50s of BRPF1/2/3=7.9/48/260 nM; Kds of BRPF1/2/3=40/210/940 nM). It also has excellent selectivity over nonclass IV BRD proteins.

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      • Nicodicosapent

        Ref: T16322
        Sizes: 25 mg, 100 mg, 50 mg, 2 mg
        From: €107.00

        Nicodicosapent (Legacy Tebubio ref. 282T16322). Nicodicosapent is a fatty acid niacin conjugate and an inhibitor of the sterol regulatory element-binding protein (SREBP), which is a key regulator of cholesterol metabolism proteins such as PCSK9, HMG-CoA reductase, ATP citrate lyase, and NPC1L1.

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      • Nigericin

        Ref: T16323
        Sizes: 25 mg
        Price Enquiry

        Nigericin (Legacy Tebubio ref. 282T16323). Nigericin, an antibiotic derived from Streptomyces hygroscopicus, acts as a K+/H+ ionophore, promoting K+/H+ exchange across mitochondrial membranes. It can activate NLRP3 and cause the release of IL-1β in a NALP3-dependent manner. Nigericin induces eryptosis, partly due to oxidative stress and ROS formation, and also causes apoptosis.

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      • Nimbolide

        Ref: T16324
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €92.00

        Nimbolide (Legacy Tebubio ref. 282T16324). Nimbolide suppresses CDK4/CDK6 kinase activity. Nimbolide inhibits the NF-κB, Wnt, PI3K-Akt, MAPK, and JAK-STAT signaling pathways. Nimbolide causes apoptosis through the inactivation of NF-κB. Nimbolide is a triterpene derived from the leaves and flowers of neem (Azadirachta indica L).

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      • NITD008

        Ref: T16325
        Sizes: 1 mg
        From: €197.00

        NITD008 (Legacy Tebubio ref. 282T16325). NITD008 (7-Deaza-2'-C-acetylene-adenosine) is a potent and selective adenosine nucleoside inhibitor.NITD008 is an adenosine nucleoside analog with broad-spectrum antiviral activity that inhibits dengue, animal cupripoxvirus, and Zika virus.

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      • Cipargamin

        Ref: T16326
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €37.00

        Cipargamin (Legacy Tebubio ref. 282T16326). Cipargamin (NITD609) is an effective antimalarial compound. It has an IC50 of appr 1 nM against P. falciparum.

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