Skip to main content
Customer Service: +351 215 842 958
Contact us
(0)
My Wishlist
(0)
My Wishlist
(0)
My WishlistContact us
Products banner

Activators & Inhibitors

Filters

    Results for Activators & Inhibitors ( 70847 )

      • NVP-2

        Ref: T16363
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €57.00

        NVP-2 (Legacy Tebubio ref. 282T16363). NVP-2 is an effective and selective ATP-competitive cyclin-dependent kinase 9 (CDK9) probe. NVP-2 induces cell apoptosis. NVP-2 inhibits CDK9/CycT activity (IC50: 0.514 nM). NVP-2 shows inhibitory effcts on CDK1/CycB, CDK2/CycA and CDK16/CycY kinases (IC50: 0.584 μM, 0.706 μM, and 0.605 μM, respectively).

        Product detail

      • Infigratinib phosphate

        Ref: T16364
        Sizes: 5 mg, 25 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €45.00

        Infigratinib phosphate (Legacy Tebubio ref. 282T16364). Infigratinib phosphate (BGJ-398 phosphate) is an effective inhibitor of the FGFR family (IC50: 0.9 nM, 1.4 nM, 1 nM, and 60 nM for FGFR1, FGFR2, FGFR3, and FGFR4, respectively).

        Product detail

      • Buparlisib Hydrochloride

        Ref: T16365
        Sizes: 2 mg
        From: €41.00

        Buparlisib Hydrochloride (Legacy Tebubio ref. 282T16365). Buparlisib Hydrochloride is an inhibitor of pan-class I PI3K (IC50: 52 nM/166 nM/116 nM/262 nM for p110α/p110β/p110δ/p110γ, respectively).

        Product detail

      • NVR 3-778

        Ref: T16366
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €58.00

        NVR 3-778 (Legacy Tebubio ref. 282T16366). NVR 3-778 is a first-in-class, orally bioavailable HBV CAM belonging to the SBA class, exhibiting anti-HBV activity.

        Product detail

      • NVS-PAK1-1

        Ref: T16367
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €50.00

        NVS-PAK1-1 (Legacy Tebubio ref. 282T16367). NVS-PAK1-1 is an effective and selective allosteric PAK1 inhibitor (IC50: 5 nM).

        Product detail

      • NVX-207

        Ref: T16368
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg
        From: €594.00

        NVX-207 (Legacy Tebubio ref. 282T16368). NVX-207 is a derivative of betulinic acid. It has anti-cancer activity.

        Product detail

      • O-Desmethyl gefitinib

        Ref: T16369
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €58.00

        O-Desmethyl gefitinib (Legacy Tebubio ref. 282T16369). O-Desmethyl gefitinib inhibits EGFR (IC50: 36 nM in subcellular assays). In human plasma, O-Desmethyl gefitinib is an active metabolite of Gefitinib. The formation of O-desmethyl gefitinib is dependent on the CYP2D6 activity.

        Product detail

      • Paroxetine hydrochloride hemihydrate

        Ref: T1636L
        Sizes: 25 mg, 100 mg, 50 mg, 500 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €35.00

        Paroxetine hydrochloride hemihydrate (Legacy Tebubio ref. 282T1636L). Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).

        Product detail

      • Deferoxamine Mesylate

        Ref: T1637
        Sizes: 1 g, 100 mg, 50 mg, 500 mg, 1 mL * 10 mM (in DMSO)
        From: €36.00

        Deferoxamine Mesylate (Legacy Tebubio ref. 282T1637). Deferoxamine Mesylate (DFOM) is an iron chelator and ferroptosis inhibitor. Deferoxamine Mesylate binds free iron into a stable complex and reduces iron accumulation. Deferoxamine Mesylate up-regulates HIF-1α levels and induces apoptosis.

        Product detail