Skip to main content
Filters

    Results for Activators & Inhibitors ( 70847 )

      • Ref: T16401
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: €46.00

        Org-12962 (Legacy Tebubio ref. 282T16401). Org-12962 is an effective and selective 5-HT2C receptor agonist pEC50: 7.01). Org-12962 shows antiaversive effects in a rat model of panic-like anxiety. Org-12962 also shows high effacy for the 5-HT2A and 5-HT2B receptors (pEC50s: 6.38 and 6.28, respectively).

        Product detail
      • Ref: T16402
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 1 mL * 10 mM (in DMSO)
        From: €45.00

        Org-26576 (Legacy Tebubio ref. 282T16402). Org-26576 is a positive allosteric modulator of the AMPA receptor.

        Product detail
      • Ref: T16403
        Sizes: 1 mg
        From: €226.00

        Org41841 (Legacy Tebubio ref. 282T16403). Org41841 is an agonist of luteinising hormone/chorionic gonadotropin receptor and thyroid stimulating hormone receptor (EC50s: 0.2 and 7.7 μM, respectively) and can be used to study hyperthyroidism.

        Product detail
      • Ref: T16404
        Sizes: 25 mg, 100 mg, 50 mg
        From: €2,747.00

        ORIC-101 (Legacy Tebubio ref. 282T16404). ORIC-101 is a highly effective and selective glucocorticoid receptor antagonist (EC50: 5.6 nM). It also has anti-cancer activity.

        Product detail
      • Ref: T16405
        Sizes: 25 mg, 100 mg, 50 mg
        From: €1,726.00

        Ornidazole diol (Legacy Tebubio ref. 282T16405). Ornidazole diol is a diol produced through ornidazole rapidly hydrolyzing in basic solutions.

        Product detail
      • Ref: T16406
        Sizes: 25 mg, 100 mg, 50 mg
        From: €781.00

        Orvepitant maleate (Legacy Tebubio ref. 282T16406). Orvepitant maleate is an effective, selective, and well-tolerated neurokinin-1 receptor (NK-1) antagonist (pKi: 10.2 for human neurokinin-1 receptor). Orvepitant maleate has the potential for depressive disorder and chronic refractory cough (CRC) treatment. Orvepitant maleate can across the blood-brain barrier.

        Product detail
      • Ref: T16407
        Sizes: 5 mg

        Osajin (Legacy Tebubio ref. 282T16407). Osajin is the major bioactive iso avone present in the fruit of Maclura pomifera. It has antitumor, antioxidant, and anti-inflammatory activities.

        Product detail
      • Ref: T16408
        Sizes: 25 mg, 100 mg, 50 mg
        From: €2,520.00

        Osanetant (Legacy Tebubio ref. 282T16408). Osanetant produces anxiolytic- and antidepressant-like effects. Osanetant is a selective NK3 receptor antagonist. It is researched for schizophrenia.

        Product detail
      • Ref: T16409
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: €39.00

        OSMI-1 (Legacy Tebubio ref. 282T16409). OSMI-1 is an O-GlcNAc transferase (OGT) inhibitor (IC50=2.7 μM) that is orally active and cell-permeable. OSMI-1 inhibits protein O-GlcNA acetylation without qualitatively altering cell-surface N- or O- linked glycans.

        Product detail