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Chemicals & Small Molecules

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    Results for Chemicals & Small Molecules ( 97587 )

      • GSK3368715 3HCl

        Ref: T22342
        Sizes: 25 mg, 100 mg, 50 mg
        From: £2,564.00

        GSK3368715 3HCl (Legacy Tebubio ref. 282T22342). GSK3368715, a potent inhibitor of type I protein arginine methyltransferases (PRMT), could inhibit PRMT1, 3, 4, 6 and 8 with Kiapp vaules ranging from 1.5 to 81 nM.

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      • HKB99

        Ref: T22343
        Sizes: 1 mg
        From: £283.00

        HKB99 (Legacy Tebubio ref. 282T22343). HKB99 is a mutant inhibitor of phosphoglycerate mutase 1 (PGAM1), which inhibits the growth and metastasis of non-small cell lung cancer.HKB99 acts synergistically with EGFR inhibitors and assists in the killing of tumors by EGFR inhibitors.HKB99 promotes oxidative stress, which induces alterations in a variety of signaling pathways.HKB99 can be used in the study of metabolism-related diseases.HKB99 can be used in the study of metabolism-related diseases.HKB99 can be used in the study of metabolism-related diseases.

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      • Icatibant Acetate

        Ref: T22344
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: £61.00

        Icatibant Acetate (Legacy Tebubio ref. 282T22344). Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.

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      • INCB054329

        Ref: T22345
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: £37.00

        INCB054329 (Legacy Tebubio ref. 282T22345). INCB054329, a structurally distinct bromodomain and extraterminal domain (BET) inhibitor, inhibits BRD2-BD1, BRD2-BD2, BRD3-BD1, BRD3-BD2, BRD4-BD1, BRD4-BD2, BRDT-BD1 and BRDT-BD2 with IC50 values of 44 nM, 5 nM, 9 nM, 1 nM, 28 nM, 3 nM, 119 nM and 63 nM respectively.

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      • Indomethacin sodium hydrate

        Ref: T22346
        Sizes: 1 g, 500 mg, 1 mL * 10 mM (in DMSO)
        From: £38.00

        Indomethacin sodium hydrate (Legacy Tebubio ref. 282T22346). Indomethacin sodium hydrate (Indometacin sodium hydrate) is an orally active, competitive and reversible COX1/2 inhibitor with potential anti-inflammatory activity in induced migraines, induced gastrointestinal injuries, and may be used in studies of increased intracranial pressure secondary to severe traumatic brain injury and rheumatoid arthritis in adults.

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      • Isonipecotic acid

        Ref: T22348
        Sizes: 1 g
        From: £28.00

        Isonipecotic acid (Legacy Tebubio ref. 282T22348). Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.

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      • JNJ-38158471

        Ref: T22349
        Sizes: 1 mg, 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 200 mg, 2 mg, 1 mL * 10 mM (in DMSO)
        From: £46.00

        JNJ-38158471 (Legacy Tebubio ref. 282T22349). JNJ-38158471 (CS-2660), a highly selective, orally available, well tolerated VEGFR2 inhibitor with IC50 of 40 nM, inhibits closely related tyrosine kinases such as Ret and Kit with IC50 of 180 nM and 500 nM.

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      • Dactolisib

        Ref: T2235
        Sizes: 25 mg, 100 mg, 50 mg, 200 mg
        From: £38.00

        Dactolisib (Legacy Tebubio ref. 282T2235). Dactolisib (BEZ235) is an orally bioavailable inhibitor of PI3K and mTOR, with IC50 values of 4 nM for p110α, 5 nM for p110γ, 7 nM for p110δ, 75 nM for p110β, and 20.7 nM for mTOR.

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      • JX06

        Ref: T22350
        Sizes: 5 mg, 25 mg, 100 mg, 50 mg, 10 mg, 1 mL * 10 mM (in DMSO)
        From: £41.00

        JX06 (Legacy Tebubio ref. 282T22350). JX06, a potent, selective and covalent PDK inhibitor, inhibits PDK1, PDK2 and PDK3 with IC50 of 49 nM, 101 nM and 313 nM respectively.

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